Home > Community > Deprotection of carboxybenzyl (Cbz) in the presence of Methyl ester?
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Aaysha Safare

Deprotection of carboxybenzyl (Cbz) in the presence of Methyl ester?

Brian Smyth  Follow

Just leave out the last step, i.e., LiOH/MeOH and you should be just fine, the Cbz group gets removed under reductive conditions which leave the methyl ester unaffected. If you lose the methyl ester, you could just add it again afterwards.

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Electricity & Electronics  Follow
) One other approach would be to use another reducing reagent for the deprotection that leaves the ester unaffected (NaBH3CN?)More
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Edwin Amhanokhai A.  Follow
I would at least not suspect esters to be very labile in Pd/C hydrogenation. While this is in principle possible, the carbamate of the Cbz will be cleaved quicker. So, I dont really see that to be a significant problem. Here are two references that look pretty similar to your problem: T. Maki, T. Tsuritani, T. Yasukata, Org. Lett., 2014, 16, 1868-1871. G. S. Vanier, Synlett, 2007, 131-135. (see More
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E. Milton Wilson  Follow
organic-chemistry.org/protectivegroups/amino/cbz-amino.htmMore
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Joe Dorety  Follow
Are you sure that reduction using Pd/C will not cleave the methyl group. As, I know t-Butyl ester is stable against reducing agent like Pd/C but I am not sure about Methyl group. any insight or reference ?More
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