Ritanserin RC10100
3 Inquiries
87051-43-2
Pharmaceutical Grade
99%
Royalchem
25kg/drum
Yes
2030-01-01
Pharmaceutical intermediates
-
Product Description
-
Seller Information
-
Inquiry History
-
DescriptionECHEMI Editorial ReferenceRitanserin is a thiazolopyrimidine that is 5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one which is substituted at position 7 by a methyl group and at position 6 by a 2-{4-[bis(4-fluorophenyl)methylidene]piperidin-1-yl}ethyl group. A potent and long-acting seratonin (5-hydroxytryptamine, 5-HT) antagonist of the subtype 5-HT2 (Ki = 0.39 nM), it is used in the treatment of a variety of disorders including anxiety, depression and schizophrenia. It has little sedative action. It has a role as a dopaminergic antagonist, a serotonergic antagonist, an antipsychotic agent, an anxiolytic drug, an antidepressant and an EC 3.4.21.26 (prolyl oligopeptidase) inhibitor. It is an organofluorine compound, a member of piperidines and a thiazolopyrimidine.|Ritanserin has been used in trials studying the treatment of Cocaine-Related Disorders.|A selective and potent serotonin-2 antagonist that is effective in the treatment of a variety of syndromes related to anxiety and depression. The drug also improves the subjective quality of sleep and decreases portal pressure.Basic Info
-
Product Name:
Ritanserin
Other Name:5H-Thiazolo[3,2-a]pyrimidin-5-one,6-[2-[4-[bis(4-fluorophenyl)methylene]-1-piperidinyl]ethyl]-7-methyl-;6-[2-[4-[Bis(4-fluorophenyl)methylene]-1-piperidinyl]ethyl]-7-methyl-5H-thiazolo[3,2-a]pyrimidin-5-one;Ritanserin;Tiserton;ZINC 00538314
CAS No.:87051-43-2
Molecular Formula:C27H25F2N3OS
InChIKeys:InChIKey=JUQLTPCYUFPYKE-UHFFFAOYSA-N
Molecular Weight:477.57
Exact Mass:477.57
UNII:145TFV465S
NSC Number:758470
DSSTox ID:DTXSID9042594
Categories:
Characteristics-
PSA:
65.85000
XLogP3:5.42090
Density:1.30±0.1 g/cm3
Melting Point:145.5 °C
Boiling Point:618.7±65.0 °C(Predicted)
Flash Point:328ºC
Refractive Index:1.646
Water Solubility:12.2 [ug/mL]
Storage Conditions:Store at +4ºC
Toxicity:LD50 in male, female mice, rats, dogs (mg/kg): 28.2, 28.2, 20.0, 22.2, 24.1, 33.2 i.v.; 626, 993, 956, 515, ~1280, 640-1280 orally (Awouters)
PKA:7.74±0.20
Collision Cross Section:220.7 Ų [M+H]+ [CCS Type: TW, Method: calibrated with polyalanine and drug standards]
-
-
Seller Information
-
Business Type:
Trader
-
Main Products:
Pharmaceutical intermediates
-
Location:
Room 336, Building 7, No. 177 Xingqiao North Road, Xingqiao Street, Linping District, Hangzhou
-
Payment Terms:
TT against copy of documents,D/P,L/C,TT against B/L draft before shipment,100% TT in advance
-
Average lead Time:
14 days
-
Total Annual Revenue:
Less than $1 million
-
Total Employees:
Less than 5
-
Year of Establishment:
2025
-
-
Inquiry History3 Inquiries
Country Product Purchase Quantity Date Posted 
United States
Ritanserin — CAS 87051-43-2
5 G Feb 12, 2026 
Spain
Ritanserin
1 G Sep 22, 2026
Spain
Ritanserin
5 G Aug 29, 2026 Post an enquiry for this product
More from this Seller
-
-
![Zinc formaldehyde sulfoxylate 91.0%Min RC01050]( "Zinc formaldehyde sulfoxylate 91.0%Min RC01050")
-
Zinc formaldehyde sulfoxylate 91.0%Min RC01050
Industrial Grade / 91.0%
$1/KG EXW
-
-
-
![Molecular sieve 13x RC02222]( "Molecular sieve 13x RC02222")
-
Molecular sieve 13x RC02222
Industrial Grade / 99%
$1/KG EXW
-
-
-
![Betadex sulfobutyl ether sodium RC09608]( "Betadex sulfobutyl ether sodium RC09608")
-
Betadex sulfobutyl ether sodium RC09608
Food Grade / 99%
$1/KG EXW
-
-
-
![Chloroauric acid RC03981]( "Chloroauric acid RC03981")
-
Chloroauric acid RC03981
Industrial Grade / 99%
$1/KG EXW
-
-
-
![2-Methyl-4-methoxybenzenamine RC05818]( "2-Methyl-4-methoxybenzenamine RC05818")
-
2-Methyl-4-methoxybenzenamine RC05818
Industrial Grade / 99%
$1/KG EXW
-
-
-
![Cyanamide RC06398]( "Cyanamide RC06398")
-
Cyanamide RC06398
Industrial Grade / 99%
$1/KG EXW
-
