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Home > Encyclopedia > 5-Amino-2-pyrimidinecarbonitrile

5-Amino-2-pyrimidinecarbonitrile

5-Amino-2-pyrimidinecarbonitrile structure

5-Amino-2-pyrimidinecarbonitrile 

structure
  • CAS No:

    56621-93-3

  • Formula:

    C5H4N4

  • Chemical Name:

    5-Amino-2-pyrimidinecarbonitrile

  • Synonyms:

    2-Pyrimidinecarbonitrile,5-amino-;5-Amino-2-pyrimidinecarbonitrile;2-Cyano-5-pyrimidinamine;2-Cyano-5-aminopyrimidine;5-Amino-2-cyanopyrimidine

  • Categories:

    Pharmaceutical Intermediates  >  Heterocyclic Compound

Description

White to light yellow crystal powder

5-Amino-2-pyrimidinecarbonitrile Basic Attributes

120.11206

120.11

DTXSID30480851

2933599090

Characteristics

75.6

-0.54

White to light yellow crystal powder

1.3±0.1 g/cm3

230-231 °C @ Solvent: Ethanol

367.3±34.0 °C at 760 mmHg

175.9±25.7 °C

1.600

Safety Information

|Warning|H302+H312+H332 (100%): Harmful if swallowed, in contact with skin or if inhaled [Warning Acute toxicity, oral; acute toxicity, dermal; acute toxicity, inhalation]|P261, P264, P270, P271, P280, P301+P312, P302+P352, P304+P312, P304+P340, P312, P322, P330, P363, and P501|The GHS information provided by 1 company from 1 notification to the ECHA C&L Inventory.

5-Amino-2-pyrimidinecarbonitrile Use and Manufacturing

5-Amino-2-pyrimidinecarbonitrile is used in the preparation of quinazolines as aurora 2 kinase inhibitors for the treatment of breast and colorectal cancers.

Computed Properties

Molecular Weight:120.11
XLogP3:-0.4
Hydrogen Bond Donor Count:1
Hydrogen Bond Acceptor Count:4
Exact Mass:120.043596145
Monoisotopic Mass:120.043596145
Topological Polar Surface Area:75.6
Heavy Atom Count:9
Complexity:127
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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