Home > Community > Oxidation of acetophenone to benzoic acid
Upvote

29

Downvote
+ Biochemistry
+ Synthesis
Posted by
Living with Adult ADHD

Oxidation of acetophenone to benzoic acid

Alina Nasir  Follow

I'd like to clear up one issue that has not been addressed in comments, but provides a weak answer.

There are NO benzylic hydrogens in acetophenone. So it is not possible based on what the textbook tells you.

More

Upvote

VOTE

Downvote
Imasha Dewmini Perera  Follow
youve nailed one of the points I was trying to make ... why does my text fail to be self-consistent? Well, I guess I already know the answer ...More
Upvote

VOTE

Downvote
Jim Young  Follow
This may be Bayer-Villager variant, but Ive been away from teaching for awhile, and never used this reaction in my lab work, so it is not familiar to me. My intuition tells me chromic acid is not strong enough, but Id never bet my intuition against a good literature search.More
Upvote

VOTE

Downvote
Carlos Torres  Follow

From a SciFinder search, there are ~10 examples of oxidations of aryl methyl ketones resulting in a carboxylic acid using a chromium based reagent (usually dichromate but also chromium trioxide). This suggests the reaction is at least possible, although I think including it in a textbook is unwarranted.

One reaction slipped through my search that is informative (below). Notice that in the presence of a benzylic position that does contain a hydrogen, the methyl ketone is unchanged, while the other group is oxidized.

enter image description here

Taken together, it seems that chromium oxidation of an acetophenone to a carboxylic acid is slower than alkyl benzylic oxidation.

More

Upvote

VOTE

Downvote