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Saxagliptin structure

Saxagliptin structure

Saxagliptin

Saxagliptin(BMS477118) is a selective and reversible DPP4 inhibitor with IC50 of 26 nM and Ki of 1.3 nM.IC50 value: 26 nM [1]Target: DPP4in vitro: Saxagliptin has an inhibition constant Ki of 1.3 nM for DPP4 inhibition, which is 10-fold more potent than either vildagliptin or sitagliptin (another two DPP4 inhibitors) with Ki of 13 and 18 nM. In addition, Saxagliptin demonstrates greater specificity for DPP4 than for either the DPP8 or DPP9 enzymes (400- and 75- fold, respectively). The a

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ALIVUS LIFE SCIENCES LTD
United States United States

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TAPI NL B.V.
France France

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    2025-02-04 00:00:00
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    France France
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    55 Piet Heinkade 1019GM Amsterdam PAYS-BAS
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Shandong Anhong Pharmaceutical Co., Ltd.
China China

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    2009-06-01
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    China China
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    No. 29, Huayuan Street, Linyi County, Dezhou City, Shandong Province
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    91371424689490635F
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    30 million yuan
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Jiangsu Hansoh Pharmaceutical Group Co., Ltd.
China China

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    1995-07-26
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    China China
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    Lianyungang Economic and Technological Development Zone, Jiangsu Province
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    913207006083959289
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    1,000,000,000 Yuan
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Hefei Cosource Heyuan Pharmaceutical Co., Ltd.
China China

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    2006-09-08
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    China China
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    No. 358, Ganquan Road, Hefei City, Anhui Province
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Aurovitas PHARMA Taizhou Co., Ltd.
China China

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    2018-01-29
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    China China
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AstraZeneca Investment (China) Co., Ltd.
China China

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    2007-09-20
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    China China
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    No. 199, Liangjing Road, China (Shanghai) Pilot Free Trade Zone
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    91310000717881028D
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Zhejiang SUPOR Pharmaceuticals Co., Ltd.
China China

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    2002-05-30
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    China China
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    Yuedong Road, Yuecheng District, Shaoxing City, Zhejiang Province
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    9133060073990848XA
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    50 million yuan
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Lianyungang Runzhong Pharmaceutical Co., Ltd.
China China

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    2010-10-20
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    China China
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    No. 16, Jinqiao Road, Dapu Industrial Zone, Lianyungang Economic and Technological Development Zone
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Yangzhou NO.3 Pharmacitical Manufacture Co., Ltd.
China China

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    2000-12-28
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    China China
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    No. 51, Guotai Road, Yiling Town, Jiangdu District, Yangzhou City
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    91321012717489085N
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