TC-DAPK 6
315694-89-4
0.98%
2026-10-20
Coenzymes,Inhibito,Enzymes,Zymogens,Substrates,Native Microorganism Creatine Amidinohydrolase
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Product Description
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Seller Information
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Description
ProductName TC-DAPK 6 Cat No CEI-1551 Product Overview Death-associated protein kinase (DAPK) is a serine/threonine protein kinase implicated in diverse programmed cell death pathways. DAPK is a promising target protein for the treatment of ischemic diseases. TC-DAPK 6 is an oxazalone compound that acts as a potent, ATP-competitive, and highly selective death-associated protein kinase (DAPK) inhibitor (IC50 = 69 and 225 nM against DAPK1 and DAPK3, respectively, with 10 μM ATP); while exhibiting much reduced or no activity against a panel of 48 other kinases even at concentrations as high as 10 μM. CAS No 315694-89-4 Molecular Weight 276.29 Purity 0.98 Storage Store at -20°C Synonyms DAPK inhibitor Targets DAPK Molecular Formula C17H12N2O2 Chemical Name (4E)-2-[(E)-2-phenylethenyl]-4-(pyridin-3-ylmethylidene)-1,3-oxazol-5-one Solubility Soluble in DMSO > 10 mM Shipping Conditions Evaluation sample solution: ship with blue ice. All other available size: ship with RT, or blue ice upon request category Specialty Chemicals(c26) cas_num 315694-89-4 Basic Info-
Product Name:
(4Z)-2-[(E)-2-phenylethenyl]-4-(pyridin-3-ylmethylidene)-1,3-oxazol-5-one
Other Name:TC-DAPK 6;CHEMBL565286;315694-89-4;4-(pyridin-3-ylmethylene)-2-styryloxazol-5(4H)-one;MLS001001987;SCHEMBL16500470;ZINC4867554;4087AH;BDBM50299910;AKOS001425611;NE58146;NCGC00387161-01;SMR000353353;W-5342;(4Z)-4-(3-pyridylmethylene)-2-[(E)-styryl]oxazol-5-one;(4Z)-2-[(E)-2-Phenylethenyl)-4-(3-pyridinylmethylene)-5(4H)-oxazolone;(4Z)-2-[2-Phenylethenyl]-4-(pyridin-3-ylmethylidene)-1,3-oxazol-5-one;(4Z)-2-[(E)-2-phenylethenyl]-4-(pyridin-3-ylmethylidene)-4,5-dihydro-1,3-oxazol-5-one;2-(2-phenylethenyl)-4-(pyridin-3-ylmethylidene)-4,5-dihydro-1,3-oxazol-5-one
CAS No.:315694-89-4
Molecular Formula:C17H12N2O2
InChIKeys:GFGMISOSPOPSHN-NOCYUORASA-N
Molecular Weight:276.29 g/mol
Exact Mass:276.089877630 g/mol
DSSTox ID:DTXSID10420639
Categories:
Characteristics-
PSA:
51.6 Ų
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Seller Information
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Business Type:
Manufactory
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Main Products:
Coenzymes,Inhibito,Enzymes,Zymogens,Substrates,Native Microorganism Creatine Amidinohydrolase
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Location:
Shirley, New York 11967, USA
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Payment Terms:
TT against copy of documents,D/P
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Average lead Time:
15 days
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Total Annual Revenue:
$1 million-$2.5 million
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Year of Establishment:
2004
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