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1138245-13-2 Mirogabalin API powder

22 Inquiries

Unit Price:

$100/G FOB

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CAS No.:

1138245-13-2

Grade:

Pharmaceutical Grade

Content:

99%

Port:

qingdao

Brand:

Packaging:

according to your request

Price valid (until):

2028-11-29

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NATURE INDUSTRIAL LIMITED

Company Type:

Trader

Location:

Hongkong, China

Payment Terms:

TT against copy of documents,D/P,L/C,D/A,O/A,TT against B/L draft before shipment,100% TT in advance

Average Lead Time:

7 days

Qualification:

Main Products:

Weight Loss Peptide,Reta,Tirz,Sema,5 Amino 1mq,Cosmetic raw material,API,SLU-PP-332

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Product Description
Seller Information
Inquiry History

Description

Parameter Item	Description
Chemical Name	Mirogabalin
Category	Synthetic gabapentinoid (α2δ ligand), pharmaceutical raw material
Appearence	White to off-white crystalline powder
Molecular Formula	C12H19NO2
Molecular Weight	209.28500
Solubility	Freely soluble in water; soluble in methanol, ethanol, dimethyl sulfoxide
Brand	Tongze
CAS Number	1138245-13-2

Milobarin is an oral gabapentin drug developed by Daiichi Sankyo, mainly used to treat peripheral neuropathy (PNP), including diabetes peripheral neuropathy (DPN), post herpetic neuralgia (PHN) and trigeminal neuralgia (TN). The drug binds to the voltage-gated calcium channel α 2 δ -1 subunit in the nervous system and regulates it, playing a role in treating chronic neuropathic pain.

Shop High Purity Pharmaceutical Grade CAS 1138245-13-2 Mirogabalin Analgesic API-Detailed Image 1

Milo Bahrain is a novel preferentially selective α 2 δ -1 ligand with high potency and selectivity towards the α 2 δ -1 subunit of voltage sensitive calcium channel complexes in the central nervous system. Data shows that in in vitro experiments using membrane preparations derived from human and rat α 2 δ subunit expressing cells, compared to Pregabal, the dissociation rate of Milo Bahrain from α 2 δ -2 is slower than that of α 2 δ -2, especially α 2 δ -1. In addition, milobarin showed high efficiency and sustained analgesic effect in streptozotocin induced diabetes rats. Its superior analgesic effect and wider CNS safety range were attributed to its selective and slow dissociation of α 2 δ -1 compared with Pregabal.
Milobarin, as an α 2 δ -1 ligand, is used to treat pain related to diabetes peripheral neuropathy, fibromyalgia and post herpetic neuralgia. Milo Bahrain targets α 2 δ -1, an accessory protein associated with voltage sensitive calcium channel complexes in the central nervous system, which reduces calcium influx into nerve endings and thus decreases the release of various pain neurotransmitters.
Application fields:
In the field of medicine, Milo Bahrain can be used alone or in combination with trazodone or its salts, gabapentin or Pregabal to treat neuropathic pain, cardiovascular diseases and other conditions. In addition, Milo Bahrain is a natural antioxidant that can effectively neutralize free radicals and reduce their damage to the skin. Therefore, it is widely used in skincare products to protect the skin from free radical damage. It can also promote the production of collagen, increase skin elasticity and firmness, making the skin appear younger and healthier. Milo Bahrain also has anti-inflammatory and anti allergic properties, which help alleviate skin allergic reactions, reduce discomfort such as redness, swelling, and itching.
In addition to medication and skincare products, Milo Bahrain can also benefit from its antioxidant properties through dietary intake. Some foods rich in Milo Bahrain include blueberries, strawberries, pomegranates, carrots, etc. Increasing the intake of these foods appropriately can help us improve the health of our skin from the inside out.

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FAQ

Q1: Are you the manufacturer or trade company?
--We are the manufacturer in China, founded on 2011.

Q2: When will the product be shipped after payment?
--The parcel will be get ready and shipped within 1 day.

Q3: How long will it take to receive the parcel?
--3-5days for the US market; 3-7days for the others.

Q4: What can I do if I don't have the ability to clear the custom.
--We got experience after doing export for many years, so don't worry we can handle that.

Q5: Why should you buy from us not from other suppliers?
---Jinan Jianfeng Chemical Co.,Ltd is a medium-sized enterprise integrating the development, production, sales and export and import trade of chemical products. Our factory has perfect infrastructure, advanced processing technology and completed detection means.

ECHEMI Editorial Reference

Mirogabalin is a calcium channel blocker with analgesic effects. It binds to the α2δ-1 and α2δ-2 subunits of voltage-dependent Ca2+channels. Mirogabalin has potent and sustained analgesic effects (ED50= 2.5 mg/kg) in rats with diabetes induced by streptozotocin (STZ; ). Mirogabalin does not inhibit activities associated with CNS adverse effects of analgesics, such as rotarod performance (ID50= 9.4 mg/kg) or locomotor activity (ID50= 43.9 mg/kg), at its effective dose. Formulations containing mirogabalin are in clinical trials for diabetic peripheral neuropathic pain.

Basic Info

Product Name:

Mirogabalin

Other Name:

2-((1R,5S,6S)-6-(aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl)acetic acid;Mirogabalin;Asapiprant;[(1R,5S,6S)-6-(Aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl]acetic acid;A200-0700;DS5565;DS5565;A200-0700;2-[(1R,5S,6S)-6-(aminomethyl)-3-ethyl-6-bicyclo[3.2.0]hept-3-enyl]acetic acid

CAS No.:

1138245-13-2

Molecular Formula:

C12H19NO2

InChIKeys:

FTBQORVNHOIASH-CKYFFXLPSA-N

Molecular Weight:

209.28

EC Number:

202-303-5

Color/Form:

Light yellow to light brown

Categories:

Other Chemical Drugs

Characteristics

Density:

1.104±0.06 g/cm3(Predicted)

Boiling Point:

357.5±15.0 °C(Predicted)

PKA:

4.65±0.10(Predicted)

Critical Temperature & Pressure:

Store at -20°C

Seller Information

Business Type:
Trader

Main Products:
Weight Loss Peptide,Reta,Tirz,Sema,5 Amino 1mq,Cosmetic raw material,API,SLU-PP-332

Location:
Unit D01,3/F., Wong King Industrial Building,No.2 Tai Yau Street, Kowloon

Payment Terms:
TT against copy of documents,D/P,L/C,D/A,O/A,TT against B/L draft before shipment,100% TT in advance

Average lead Time:
7 days

Total Annual Revenue:
$50 million-$100 million

Total Employees:
51-100

Year of Establishment:
2012

We have more than 10 years experience in the pharmacy filed. Mainly manufactures pharmaceutical APIs,Pharmaceutical intermediate and Cosmetic raw material. Owing to the good quality and competitive price, we have a very good reputation in China's pharmaceutical circles.

In the principle of "Quality Oriented", Jianfeng passed the certification of ISO9001:2008 Quality Management System.

Our products are based on bulk, high volume, wholesale price, third party testing, certificate reporting, and bring high quality ingredients to many domestic and overseas enterprises.

"Honesty, practicality, innovation, development" are our values. Jianfeng would like to cooperate with you with high quality products and competitive price.

Inquiry History

22 Inquiries

Country	Product	Purchase Quantity	Date Posted
France	Mirogabalin Besylate	1 KG	Dec 13, 2024
Pakistan	Mirogabalin	100 KG	Sep 20, 2026
United States	Mirogabalin	1 KG	May 17, 2026
United States	Mirogabalin	1 KG	Dec 14, 2025
Sweden	Mirogabalin	1 KG	Nov 1, 2025
Pakistan	Mirogabalin	100 KG	Sep 18, 2025
Pakistan	Mirogabalin	25 KG	Aug 27, 2025
Pakistan	Mirogabalin	20 KG	Sep 8, 2026
United States	Mirogabalin	1 KG	May 16, 2026
Sweden	Mirogabalin	1 KG	Feb 1, 2026
Pakistan	Mirogabalin	100 KG	Sep 21, 2026
Pakistan	Mirogabalin	25 KG	Jun 22, 2026
Netherlands	Mirogabalin	500 G	Nov 29, 2025
Pakistan	MIROGABALINE	5 KG	Nov 3, 2025
Pakistan	MIROGABALIN	100 KG	Sep 22, 2025
Pakistan	MIROGABALIN	1 MT	Jun 30, 2025
Pakistan	Mirogabalin	200 G	Feb 27, 2025
Pakistan	Mirogabalin	5 G	Feb 27, 2025
Pakistan	Mirogabalin	50 G	Feb 25, 2025
Pakistan	MIROGABALIN	0.2 KG	Oct 25, 2024

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1138245-13-2 Mirogabalin API powder

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