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Factory Supply High Quality Mirogabalin Besylate CAS 1138245-21-2

18 Inquiries

Unit Price:

$1000/G FOB

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CAS No.:

1138245-21-2

Grade:

Pharmaceutical Grade

Content:

99%

Port:

qingdao

Brand:

Packaging:

according to your request

Price valid (until):

2029-12-27

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NATURE INDUSTRIAL LIMITED

Company Type:

Trader

Location:

Hongkong, China

Payment Terms:

TT against copy of documents,D/P,L/C,D/A,O/A,TT against B/L draft before shipment,100% TT in advance

Average Lead Time:

7 days

Qualification:

Main Products:

Weight Loss Peptide,Reta,Tirz,Sema,5 Amino 1mq,Cosmetic raw material,API,SLU-PP-332

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Product Description
Seller Information
Inquiry History

Description

Product Description

Item	Mirogabalin Besylate
Storage	Store at -20°C
Appearance	Powder
MOQ	10Kg
Pakage	25Kg/Bag
Sample	Available

Quick Details:

CAS No.: 1138245-21-2

Place of Origin: China (Mainland)
Brand Name: JINLAN PHARM
We recommend T/T or Escrow , D/P,D/A, Western Union or PayPal are also acceptable!

CAS No.	1138245-21-2
Place of Origin:	China (Mainland)
Brand Name:	JINLAN PHARM

Mirogabalin Besylate: Efficacy and Clinical Functions

Mirogabalin besylate is a novel, centrally acting alpha-2-delta ligand, structurally and pharmacologically related to gabapentinoids, with potent analgesic and anxiolytic properties. It selectively binds to voltage-gated calcium channel α2δ subunits in the central nervous system, reducing excessive calcium influx and inhibiting the release of excitatory neurotransmitters such as glutamate and substance P, thereby alleviating neuropathic pain and anxiety.

Clinically, it is primarily used to treat peripheral neuropathic pain, including diabetic peripheral neuropathy and postherpetic neuralgia, effectively relieving spontaneous pain, hyperalgesia, and allodynia. It also demonstrates reliable efficacy in generalized anxiety disorder by modulating abnormal neuronal excitability, improving emotional tension, restlessness, and physical anxiety symptoms.

Compared with similar agents, mirogabalin besylate shows higher binding affinity and longer duration of action, allowing stable symptom control with relatively low dosing frequency. It is generally well tolerated, with mild and transient adverse effects, supporting its role as a valuable therapeutic option for chronic neuropathic pain and anxiety disorders.

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FAQ

Q1: Are you the manufacturer or trade company?
--We are the manufacturer in China, founded on 2011.

Q2: When will the product be shipped after payment?
--The parcel will be get ready and shipped within 1 day.

Q3: How long will it take to receive the parcel?
--3-5days for the US market; 3-7days for the others.

Q4: What can I do if I don't have the ability to clear the custom.
--We got experience after doing export for many years, so don't worry we can handle that.

Q5: Why should you buy from us not from other suppliers?
---Jinan Jianfeng Chemical Co.,Ltd is a medium-sized enterprise integrating the development, production, sales and export and import trade of chemical products. Our factory has perfect infrastructure, advanced processing technology and completed detection means.

ECHEMI Editorial Reference

Mirogabalin (DS-5565) is a drug developed by Daiichi Sankyo and related to drugs such as gabapentin and pregabalin. Similarly to these drugs, mirogabalin binds to the α2δ calcium channels (1 and 2), but with significantly higher potency than pregabalin. It has shown promising results in Phase II clinical trials for the treatment of diabetic peripheral neuropathic pain, and is currently in Phase III trials.
Mirogabalin besylate (mirogabalin, Tarlige) is a gabapentinoid therapy developed by Daiichi Sankyo, which is approved in Japan for the treatment of postherpetic neuralgia and painful diabetic peripheral neuropathy. Mirogabalin has a potent pain-modulating effect with a unique high affinity and prolonged dissociation rate for the a2delta-1 subunit of voltage-gated calcium (Ca2+) channels (VGCCs) on the dorsal root ganglion resulting in more sustained analgesia compared with traditional gabapentinoids[1].

Basic Info

Product Name:

Mirogabalin besylate

Other Name:

Mirogabalin besylate;Mirogabalin besylat;Mirogabalin Besilate;MIROGABALIN BENZENESULFONIC ACID;((1R,5S,6S)-6-(carboxymethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl)methanaminium benzenesulfonate;[(1R,5S,6S)-6-(Aminomethyl)-3-ethylbicyclo[3.2.0] hept-3-en-6-yl]acetic acid benzenesulfonate;2-((1R,5S,6S)-6-(aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl)acetic acid compound with benzenesulfonic acid (1:1);Mirogabalin Besylate 10928

CAS No.:

1138245-21-2

Molecular Formula:

C18H25NO5S

InChIKeys:

OKJXJRVWXYRSAN-QWGAVYBYNA-N

Molecular Weight:

367.46

Exact Mass:

367.145

Color/Form:

White to off-white

Categories:

Other Chemical Drugs

Characteristics

PSA:

126.07

XLogP3:

4.4968

Critical Temperature & Pressure:

Store at -20°C

Seller Information

Business Type:
Trader

Main Products:
Weight Loss Peptide,Reta,Tirz,Sema,5 Amino 1mq,Cosmetic raw material,API,SLU-PP-332

Location:
Unit D01,3/F., Wong King Industrial Building,No.2 Tai Yau Street, Kowloon

Payment Terms:
TT against copy of documents,D/P,L/C,D/A,O/A,TT against B/L draft before shipment,100% TT in advance

Average lead Time:
7 days

Total Annual Revenue:
$50 million-$100 million

Total Employees:
51-100

Year of Establishment:
2012

We have more than 10 years experience in the pharmacy filed. Mainly manufactures pharmaceutical APIs,Pharmaceutical intermediate and Cosmetic raw material. Owing to the good quality and competitive price, we have a very good reputation in China's pharmaceutical circles.

In the principle of "Quality Oriented", Jianfeng passed the certification of ISO9001:2008 Quality Management System.

Our products are based on bulk, high volume, wholesale price, third party testing, certificate reporting, and bring high quality ingredients to many domestic and overseas enterprises.

"Honesty, practicality, innovation, development" are our values. Jianfeng would like to cooperate with you with high quality products and competitive price.

Inquiry History

18 Inquiries

Country	Product	Purchase Quantity	Date Posted
United Kingdom	Factory Supply High Quality Mirogabalin Besylate CAS 1138245-21-2 white powder HHD HHD	100 G	Oct 16, 2023
Pakistan	MIROGABALIN BESYLATE	350 G	Feb 10, 2026
Pakistan	Mirogabalin Besilate	1 MT	Jul 30, 2025
Pakistan	MIROGABALIN BESYLATE	1 MT	Jul 11, 2025
Pakistan	Mirogabalin Besylate	700 G	Oct 10, 2023
Pakistan	Mirogabalin Besylate	700 G	Sep 27, 2023
Egypt	Mirogabalin Besylate	250 KG	Apr 15, 2026
Pakistan	MIROGABALIN BESYLATE	1 MT	Mar 7, 2025
Bangladesh	Mirogabalin Besylate	1 KG	Nov 28, 2024
Bangladesh	Mirogabalin Besylate	100 KG	Nov 19, 2024
Pakistan	Mirogabalin Besylate	700 G	Sep 27, 2023
Pakistan	Mirogabalin Besylate	10 KG	Sep 4, 2026
Pakistan	Microgabalin Besylate	250 G	Aug 19, 2025
Pakistan	MIROGABLIN BESYLATE	350 G	Feb 10, 2025
Pakistan	MIROGABALIN BESYLATE	100 KG	Oct 31, 2024
Pakistan	Mirogabalin Besylate	1 KG	Jul 19, 2024
Pakistan	Mirogabalin Besylate	1 KG	Sep 27, 2023
Pakistan	Mirogabalin besylate	700 G	Sep 27, 2023

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Factory Supply High Quality Mirogabalin Besylate CAS 1138245-21-2

Product Description

Seller Information

Inquiry History

Mirogabalin Besylate: Efficacy and Clinical Functions

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