B-(3-Ethoxy-4-fluorophenyl)boronic acid

To a solution of 9A (3.86 g, 17.6 mmol) in THF (60 mL) at -78° C. was added n-BuLi (1.6 M in hexanes, 14.3 mL, 22.8 mmol). The mixture was stirred at -78° C. for 40 min before trimethyl borate (3.63 mL, 33 mmol) was added. The reaction was left stirring from -78° C. to rt over 4 h. It was quenched with 1.0 N HCl (40 mL), extracted with EtOAc, washed with brine and dried over NaTo a solution of 64B (3.86 g, 17.6 mmol) in THF (60 mL) at -78° C. was added n-BuLi (1.6 M in hexanes, 14.3 mL, 22.8 mmol). The mixture was stirred at -78° C. for 40 min before trimethyl borate (3.63 mL, 33 mmol) was added. The reaction was left stirring from -78° C. to rt over 4 h. It was quenched with 1.0 N HCl (40 mL), extracted with EtOAc, washed with brine and dried over Na

suzuki reaction

Molecular Weight:183.97
Hydrogen Bond Donor Count:2
Hydrogen Bond Acceptor Count:4
Rotatable Bond Count:3
Exact Mass:184.0707025
Monoisotopic Mass:184.0707025
Topological Polar Surface Area:49.7
Heavy Atom Count:13
Complexity:156
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes