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Bemitradine

Bemitradine structure

Bemitradine 

structure
  • CAS No:

    88133-11-3

  • Formula:

    C15H17N5O

  • Chemical Name:

    Bemitradine

  • Synonyms:

    [1,2,4]Triazolo[1,5-c]pyrimidin-5-amine,8-(2-ethoxyethyl)-7-phenyl-;8-(2-Ethoxyethyl)-7-phenyl[1,2,4]triazolo[1,5-c]pyrimidin-5-amine;SC 33643;Bemitradine

Description

Bemitradine is a triazolopyrimidine derivative diuretic. Bemitradine has thiazide-like actions and is a renal vasodilator. Due to its non-genotoxic carcinogenicity, clinical development for this agent has stopped.

Bemitradine Basic Attributes

283.333

283.33

LT9004D9N0

DTXSID7020132

C77556

2933990090

Characteristics

78.3

1.88260

1.31±0.1 g/cm3(Predicted)

Drug Information

8-(2-ethoxyethyl)-7-phenyl-1,2,4-triazolo-1,5c-pyrimidine-5-amine

Bemitradine Use and Manufacturing

Antihypertensive; diuretic.

Computed Properties

Molecular Weight:283.33
XLogP3:1.9
Hydrogen Bond Donor Count:1
Hydrogen Bond Acceptor Count:5
Rotatable Bond Count:5
Exact Mass:283.14331018
Monoisotopic Mass:283.14331018
Topological Polar Surface Area:78.3
Heavy Atom Count:21
Complexity:323
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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