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Cimetidine sulfoxide

Cimetidine sulfoxide structure

Cimetidine sulfoxide 

structure
  • CAS No:

    54237-72-8

  • Formula:

    C10H16N6OS

  • Chemical Name:

    Cimetidine sulfoxide

  • Synonyms:

    Guanidine,N-cyano-N′-methyl-N′′-[2-[[(4-methyl-1H-imidazol-5-yl)methyl]sulfinyl]ethyl]-;Guanidine,N-cyano-N′-methyl-N′′-[2-[[(5-methyl-1H-imidazol-4-yl)methyl]sulfinyl]ethyl]-;N-Cyano-N′-methyl-N′′-[2-[[(4-methyl-1H-imidazol-5-yl)methyl]sulfinyl]ethyl]guanidine;Cimetidine sulfoxide;(±)-Cimetidine S-oxide;SKF 92452;1-Cyano-2-methyl-3-[2-[(5-methyl-1H-imidazol-4-yl)methylsulfinyl]ethyl]guanidine;151378-35-7

Description

Cimetidine S-oxide is a sulfoxide. It derives from a cimetidine.

Cimetidine sulfoxide Basic Attributes

268.339

268.34

Characteristics

125

-1.1

1.39±0.1 g/cm3(Predicted)

608.6ºC at 760mmHg

321.8ºC

1.665

Drug Information

1-cyano-2-methyl-3-(2-(((4-methyl-1H-imidazol-5-yl)methyl)sulfinyl)ethyl)guanidine

Cimetidine sulfoxide Use and Manufacturing

Cimetidine Sulfoxide is a metabolite of the H2-receptor antagonist Cimetidine (C441650). Cimetidine Sulfoxide is detected in the blood and urine of patients with kidney diseases.

Computed Properties

Molecular Weight:268.34
XLogP3:-1.1
Hydrogen Bond Donor Count:3
Hydrogen Bond Acceptor Count:5
Rotatable Bond Count:7
Exact Mass:268.11063033
Monoisotopic Mass:268.11063033
Topological Polar Surface Area:125
Heavy Atom Count:18
Complexity:363
Undefined Atom Stereocenter Count:1
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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