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Cilostamide

Cilostamide structure

Cilostamide 

structure
  • CAS No:

    68550-75-4

  • Formula:

    C20H26N2O3

  • Chemical Name:

    Cilostamide

  • Synonyms:

    Butanamide,N-cyclohexyl-4-[(1,2-dihydro-2-oxo-6-quinolinyl)oxy]-N-methyl-;N-Cyclohexyl-4-[(1,2-dihydro-2-oxo-6-quinolinyl)oxy]-N-methylbutanamide;Cilostamide;OPC 3689

  • Categories:

    Cosmetic Ingredient  >  Skin Protecting

Description

Cilostamide is a selective and potent PDE3 inhibitor, with IC50s of 27 nM and 50 nM for PDE3A and PDE3B, respectively, and has antithrombotic and anti-intimal hyperplastic activity.


N-cyclohexyl-N-methyl-4-[(2-oxo-1H-quinolin-6-yl)oxy]butanamide is a member of quinolines.

Cilostamide Basic Attributes

342.43

342.43

45S5605Q18

DTXSID3045140

Characteristics

58.6

2.70

1.2±0.1 g/cm3

186-188 °C @ Solvent: Methanol, Water

594.3±50.0 °C at 760 mmHg

313.2±30.1 °C

1.586

0-6°C

Safety Information

III

6.1(b)

3249

3

Drug Information

Compounds which inhibit or antagonize the biosynthesis or actions of phosphodiesterases. (See all compounds classified as Phosphodiesterase Inhibitors.)|Drugs or agents which antagonize or impair any mechanism leading to blood platelet aggregation, whether during the phases of activation and shape change or following the dense-granule release reaction and stimulation of the prostaglandin-thromboxane system. (See all compounds classified as Platelet Aggregation Inhibitors.)

cilostamide

Cilostamide Use and Manufacturing

Serotonin receptor ligand

Computed Properties

Molecular Weight:342.4
XLogP3:2.9
Hydrogen Bond Donor Count:1
Hydrogen Bond Acceptor Count:3
Rotatable Bond Count:6
Exact Mass:342.19434270
Monoisotopic Mass:342.19434270
Topological Polar Surface Area:58.6
Heavy Atom Count:25
Complexity:499
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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