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Desmethylmianserin

Desmethylmianserin structure

Desmethylmianserin 

structure
  • CAS No:

    71936-92-0

  • Formula:

    C17H18N2

  • Chemical Name:

    Desmethylmianserin

  • Synonyms:

    Dibenzo[c,f]pyrazino[1,2-a]azepine,1,2,3,4,10,14b-hexahydro-;1,2,3,4,10,14b-Hexahydrodibenzo[c,f]pyrazino[1,2-a]azepine;Demethylmianserin;Desmethylmianserin;Normianserin;(±)-Demethylmianserin;Normianserine;N-Desmethylmianserin;77862-25-0

Description

Off-White Solid

Desmethylmianserin Basic Attributes

250.343

250.34

615-697-2

Characteristics

15.3

2.9

87-89°C

Refrigerator

Drug Information

Normianserin is a known transformation product of Mianserin.

Desmethylmianserin is a known human metabolite of Mianserine.

1,2,3,4,10,14b-hexahydrodibenzo(c,f)pyrazino(1,2-a)azepine

Desmethylmianserin Use and Manufacturing

Uses

The active metabolites of Miansein (M341500) in plasma, an antidepressant

Pharmaceuticals -> Transformation products

Computed Properties

Molecular Weight:250.34
XLogP3:2.9
Hydrogen Bond Donor Count:1
Hydrogen Bond Acceptor Count:2
Exact Mass:250.146998583
Monoisotopic Mass:250.146998583
Topological Polar Surface Area:15.3
Heavy Atom Count:19
Complexity:316
Undefined Atom Stereocenter Count:1
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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