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Darodipine

Darodipine structure

Darodipine 

structure
  • CAS No:

    72803-02-2

  • Formula:

    C19H21N3O5

  • Chemical Name:

    Darodipine

  • Synonyms:

    3,5-Pyridinedicarboxylic acid,4-(2,1,3-benzoxadiazol-4-yl)-1,4-dihydro-2,6-dimethyl-,3,5-diethyl ester;3,5-Pyridinedicarboxylic acid,4-(4-benzofurazanyl)-1,4-dihydro-2,6-dimethyl-,diethyl ester;3,5-Pyridinedicarboxylic acid,4-(2,1,3-benzoxadiazol-4-yl)-1,4-dihydro-2,6-dimethyl-,diethyl ester;2,1,3-Benzoxadiazole,3,5-pyridinedicarboxylic acid deriv.;PY 108-068;PY 108068;Darodipine

Description

Darodipine (PY 108-068, PY-108068) is a potent calcium channel antagonist.


Darodipine is a calcium channel blocker.

Darodipine Basic Attributes

371.393

371.39

N4AL7X96GL

DTXSID90223125

Characteristics

104

2.91260

1.251g/cm3

507.3ºC at 760 mmHg

260.6ºC

1.566

Drug Information

A class of drugs that act by selective inhibition of calcium influx through cellular membranes. (See all compounds classified as Calcium Channel Blockers.)

darodipine

Darodipine Use and Manufacturing

Antihypertensive; bronchodilator; vasodilator.

Computed Properties

Molecular Weight:371.4
XLogP3:4.2
Hydrogen Bond Donor Count:1
Hydrogen Bond Acceptor Count:8
Rotatable Bond Count:7
Exact Mass:371.14812078
Monoisotopic Mass:371.14812078
Topological Polar Surface Area:104
Heavy Atom Count:27
Complexity:632
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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