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Demegestone

Demegestone structure

Demegestone 

structure
  • CAS No:

    10116-22-0

  • Formula:

    C21H28O2

  • Chemical Name:

    Demegestone

  • Synonyms:

    19-Norpregna-4,9-diene-3,20-dione,17-methyl-;17-Methyl-19-norpregna-4,9-diene-3,20-dione;Demegestone;R 2453;Lutionex;RU 2453;NSC 118189

Description

Demegestone is a 20-oxo steroid.|Demegestone is a progesterone receptor agonist that was previously used to treat luteal insufficiency. It was previously marketed in France as Lutionex, but has since been discontinued.

Demegestone Basic Attributes

312.453

312.45

233-320-6

6E89AM91SZ

G - Genito urinary system and sex hormones

Characteristics

34.1

4.78770

1.11g/cm3

106 °C

475.5ºC at 760mmHg

176.6ºC

1.557

3.29E-09mmHg at 25°C

D -275° (c = 0.5 in ethanol)

Drug Information

17 alpha-methyl-19-norprogesterone

Computed Properties

Molecular Weight:312.4
XLogP3:2.8
Hydrogen Bond Acceptor Count:2
Rotatable Bond Count:1
Exact Mass:312.208930132
Monoisotopic Mass:312.208930132
Topological Polar Surface Area:34.1
Heavy Atom Count:23
Complexity:653
Defined Atom Stereocenter Count:4
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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