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Pafuramidine

Pafuramidine structure

Pafuramidine 

structure
  • CAS No:

    186953-56-0

  • Formula:

    C20H20N4O3

  • Chemical Name:

    Pafuramidine

  • Synonyms:

    Benzenecarboximidamide,4,4′-(2,5-furandiyl)bis[N-methoxy-;4,4′-(2,5-Furandiyl)bis[N-methoxybenzenecarboximidamide];2,5-Bis(4-amidinophenyl)furan-bis-O-methylamidoxime;Pafuramidine

Pafuramidine Basic Attributes

364.4

364.40

Characteristics

108 Ų

1.25

192.5-193 °C

457.7±55.0 °C(Predicted)

6.01±0.50

Drug Information

Agents destructive to the protozoal organisms belonging to the suborder TRYPANOSOMATINA. (See all compounds classified as Trypanocidal Agents.)

2,5-bis(4-amidinophenyl)furan-bis-O-methylamidoxime

Pafuramidine Use and Manufacturing

Treatment of malaria, African sleeping sickness, and pneumocystis pneumonia.

Computed Properties

Molecular Weight:364.4
XLogP3:3.2
Hydrogen Bond Donor Count:2
Hydrogen Bond Acceptor Count:5
Rotatable Bond Count:6
Exact Mass:364.15354051
Monoisotopic Mass:364.15354051
Topological Polar Surface Area:108
Heavy Atom Count:27
Complexity:477
Undefined Bond Stereocenter Count:2
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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