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Home > Encyclopedia > 16-Hydroxytriptolide

16-Hydroxytriptolide

16-Hydroxytriptolide structure

16-Hydroxytriptolide 

structure
  • CAS No:

    139713-80-7

  • Formula:

    C20H24O7

  • Chemical Name:

    16-Hydroxytriptolide

  • Synonyms:

    Trisoxireno[4b,5:6,7:8a,9]phenanthro[1,2-c]furan-1(3H)-one,3b,4,4a,6,6a,7a,7b,8b,9,10-decahydro-6-hydroxy-6a-[(1S)-2-hydroxy-1-methylethyl]-,(3bS,4aS,5aS,6R,6aR,7aS,7bS,8aS,8bS)-;Triptolide,16-hydroxy-,(15S)-;(3bS,4aS,5aS,6R,6aR,7aS,7bS,8aS,8bS)-3b,4,4a,6,6a,7a,7b,8b,9,10-Decahydro-6-hydroxy-6a-[(1S)-2-hydroxy-1-methylethyl]trisoxireno[4b,5:6,7:8a,9]phenanthro[1,2-c]furan-1(3H)-one;(15S)-16-Hydroxytriptolide;16-Hydroxytriptolide;Trisoxireno[4b,5:6,7:8a,9]phenanthro[1,2-c]furan-1(3H)-one,3b,4,4a,6,6a,7a,7b,8b,9,10-decahydro-6-hydroxy-6a-(2-hydroxy-1-methylethyl)-,[3bS-[3bα,4aα,5aR*,6β,6aβ(R*),7aβ,7bα,8aR*,8bα]]-;16-Hydroxytryptolide;139601-38-0

Description

16-hydroxytriptolide is a tetracyclic diterpenoid with formula C20H24O7, originally isolated from the roots and leaves of Tripterygium wilfordii. It has a role as a plant metabolite, a rat metabolite and a xenobiotic metabolite. It is a gamma-lactone, an epoxide, a secondary alcohol, a tetracyclic diterpenoid, a primary alcohol and a diol.

16-Hydroxytriptolide Basic Attributes

376.40000

376.40

Characteristics

104.35000

0.07550

1.56g/cm3

232-233.5 °C

659.7ºC at 760mmHg

241.8ºC

1.67

3.31E-20mmHg at 25°C

Drug Information

16-hydroxytriptolide

Computed Properties

Molecular Weight:376.4
XLogP3:-1
Hydrogen Bond Donor Count:2
Hydrogen Bond Acceptor Count:7
Rotatable Bond Count:2
Exact Mass:376.15220310
Monoisotopic Mass:376.15220310
Topological Polar Surface Area:104
Heavy Atom Count:27
Complexity:838
Defined Atom Stereocenter Count:10
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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