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Amdoxovir

Amdoxovir structure

Amdoxovir 

structure
  • CAS No:

    145514-04-1

  • Formula:

    C9H12N6O3

  • Chemical Name:

    Amdoxovir

  • Synonyms:

    1,3-Dioxolane-2-methanol,4-(2,6-diamino-9H-purin-9-yl)-,(2R,4R)-;1,3-Dioxolane-2-methanol,4-(2,6-diamino-9H-purin-9-yl)-,(2R-cis)-;(2R,4R)-4-(2,6-Diamino-9H-purin-9-yl)-1,3-dioxolane-2-methanol;DAPD;β-D-2,6-Diaminopurine-dioxolane;Amdoxovir;(-)-DAPD

Description

Amdoxovir is a nucleoside reverse transcriptase inhibitor prodrug analog of guanosine.

Amdoxovir Basic Attributes

252.23 g/mol

252.23

54I81H0M9C

C76927

Characteristics

134 Ų

237-239 °C @ Solvent: Ethanol

Drug Information

Investigated for use/treatment in HIV infection and acquired immune deficiency syndrome (AIDS) and aids-related infections.

2,6-diaminopurine dioxolane

Computed Properties

Molecular Weight:252.23
XLogP3:-1.2
Hydrogen Bond Donor Count:3
Hydrogen Bond Acceptor Count:8
Rotatable Bond Count:2
Exact Mass:252.09708827
Monoisotopic Mass:252.09708827
Topological Polar Surface Area:134
Heavy Atom Count:18
Complexity:308
Defined Atom Stereocenter Count:2
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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