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Home > Encyclopedia > Hydroxyphenobarbital

Hydroxyphenobarbital

Hydroxyphenobarbital structure

Hydroxyphenobarbital 

structure
  • CAS No:

    379-34-0

  • Formula:

    C12H12N2O4

  • Chemical Name:

    Hydroxyphenobarbital

  • Synonyms:

    2,4,6(1H,3H,5H)-Pyrimidinetrione,5-ethyl-5-(4-hydroxyphenyl)-;Barbituric acid,5-ethyl-5-(p-hydroxyphenyl)-;5-Ethyl-5-(4-hydroxyphenyl)-2,4,6(1H,3H,5H)-pyrimidinetrione;p-Hydroxyphenobarbital;Hydroxyphenobarbital;p-Hydroxyphenobarbitone;5-Ethyl-5-(4-hydroxyphenyl)barbituric acid;4-Hydroxyphenobarbital;5-(p-Hydroxyphenyl)-5-ethylbarbituric acid;5-Ethyl-5-(p-hydroxyphenyl)barbituric acid;NSC 159266

Description

Off-White to Pale Yellow Solid


4-Hydroxyphenobarbital is a member of barbiturates.

Hydroxyphenobarbital Basic Attributes

248.238

248.23

206-831-7

RF9R6T1NUN

159266

DTXSID20191328

2933540000

Characteristics

95.5

1.06360

1.33g/cm3

218-220ºC

1.568

Drug Information

P-Hydroxyphenobarbital has known human metabolites that include (2S,3S,4S,5R)-6-[4-(5-ethyl-2,4,6-trioxo-1,3-diazinan-5-yl)phenoxy]-3,4,5-trihydroxyoxane-2-carboxylic acid and 4-(5-Ethyl-2,4,6-trioxohexahydropyrimidin-5-yl)phenyl hydrogen sulfate.

4-hydroxyphenobarbital

Hydroxyphenobarbital Use and Manufacturing

A metabolite of Phenobarbital

Computed Properties

Molecular Weight:248.23
XLogP3:1.1
Hydrogen Bond Donor Count:3
Hydrogen Bond Acceptor Count:4
Rotatable Bond Count:2
Exact Mass:248.07970687
Monoisotopic Mass:248.07970687
Topological Polar Surface Area:95.5
Heavy Atom Count:18
Complexity:366
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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