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Ramifenazone

Ramifenazone structure

Ramifenazone 

structure
  • CAS No:

    3615-24-5

  • Formula:

    C14H19N3O

  • Chemical Name:

    Ramifenazone

  • Synonyms:

    3H-Pyrazol-3-one,1,2-dihydro-1,5-dimethyl-4-[(1-methylethyl)amino]-2-phenyl-;Antipyrine,4-(isopropylamino)-;1,2-Dihydro-1,5-dimethyl-4-[(1-methylethyl)amino]-2-phenyl-3H-pyrazol-3-one;Isopropylaminoantipyrine;Isopropylaminophenazone;1-Phenyl-2,3-dimethyl-4-(isopropylamino)-2-pyrazolin-5-one;Isopyrine;Isopyrin;4-(Isopropylamino)antipyrine;4-Isopropylamino-2,3-dimethyl-1-phenyl-3-pyrazolin-5-one;1-Phenyl-2,3-dimethyl-4-isopropylaminopyrazolone;4-Monoisopropylamino-1-phenyl-2,3-dimethyl-5-pyrazolone;Isopirina;4-(Isopropylamino)phenazone;Ramifenazone;1,5-Dimethyl-2-phenyl-4-(propan-2-ylamino)pyrazol-3-one;1,5-Dimethyl-2-phenyl-4-[(propan-2-yl)amino]-2,3-dihydro-1H-pyrazol-3-one;2044-80-6

Description

Ramifenazone is a nonsteroidal anti-inflammatory drug.


1,5-dimethyl-2-phenyl-4-(propan-2-ylamino)-3-pyrazolone is a ring assembly and a member of pyrazoles.

Ramifenazone Basic Attributes

245.326

245.32

222-791-3

GKH2KOV2RF

DTXSID1045906

2933199090

Characteristics

35.6

0.90

1.1±0.1 g/cm3

80 °C

348.5±45.0 °C at 760 mmHg

164.6±28.7 °C

1.595

LD50 in mice (mg/kg): 843 i.p.; 1070 orally (Tubaro)

156.5 Ų [M+H]+ [CCS Type: TW, Method: calibrated with polyalanine and drug standards]

Drug Information

ramifenazone

Ramifenazone Use and Manufacturing

Uses

analgesic, antipyretic, antiinflammatory

Pharmaceuticals

Computed Properties

Molecular Weight:245.32
XLogP3:1.6
Hydrogen Bond Donor Count:1
Hydrogen Bond Acceptor Count:3
Rotatable Bond Count:3
Exact Mass:245.152812238
Monoisotopic Mass:245.152812238
Topological Polar Surface Area:35.6
Heavy Atom Count:18
Complexity:356
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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