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Pamaquine

Pamaquine structure

Pamaquine 

structure
  • CAS No:

    491-92-9

  • Formula:

    C19H29N3O

  • Chemical Name:

    Pamaquine

  • Synonyms:

    1,4-Pentanediamine,N1,N1-diethyl-N4-(6-methoxy-8-quinolinyl)-;Quinoline,8-[[4-(diethylamino)-1-methylbutyl]amino]-6-methoxy-;N1,N1-Diethyl-N4-(6-methoxy-8-quinolinyl)-1,4-pentanediamine;6-Methoxy-8-(1-methyl-4-diethylamino)butylaminoquinoline;Pamaquin;Pamaquine;Plasmochin;Plasmocide;Praequine;Prequine;Plasmoquine;Plasmoquin;Gamefar;Beprochine;Aminoquin;Quipenyl;NSC 167382

Description

primaquine (5, see Malaria)shows great promise against this protozoan in clinical trials when administered for prophylaxis or for therapy in mild to moderately severe pneumocystis pneumonia. Either drug alone is not effective.


Pamaquine is an aminoquinoline.

Pamaquine Basic Attributes

315.461

315.45

167382

Characteristics

37.4

4.1

1.028 g/cm3 @ Temp: 31 °C

<25 °C

188 °C

Drug Information

8-((4-(diethylamino)-1-methylbutyl)amino)-6-methoxyquinoline

Computed Properties

Molecular Weight:315.5
XLogP3:4.1
Hydrogen Bond Donor Count:1
Hydrogen Bond Acceptor Count:4
Rotatable Bond Count:9
Exact Mass:315.231062557
Monoisotopic Mass:315.231062557
Topological Polar Surface Area:37.4
Heavy Atom Count:23
Complexity:322
Undefined Atom Stereocenter Count:1
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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