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Home > Encyclopedia > 3-Amino-N-(aminoiminomethyl)-6-chloro-5-(methylpropylamino)-2-pyrazinecarboxamide

3-Amino-N-(aminoiminomethyl)-6-chloro-5-(methylpropylamino)-2-pyrazinecarboxamide

3-Amino-N-(aminoiminomethyl)-6-chloro-5-(methylpropylamino)-2-pyrazinecarboxamide structure

3-Amino-N-(aminoiminomethyl)-6-chloro-5-(methylpropylamino)-2-pyrazinecarboxamide 

structure
  • CAS No:

    1151-75-3

  • Formula:

    C10H16ClN7O

  • Chemical Name:

    3-Amino-N-(aminoiminomethyl)-6-chloro-5-(methylpropylamino)-2-pyrazinecarboxamide

  • Synonyms:

    2-Pyrazinecarboxamide,3-amino-N-(aminoiminomethyl)-6-chloro-5-(methylpropylamino)-;Pyrazinecarboxamide,N-amidino-3-amino-6-chloro-5-(methylpropylamino)-;Pyrazinecarboxamide,3-amino-N-(aminoiminomethyl)-6-chloro-5-(methylpropylamino)-;3-Amino-N-(aminoiminomethyl)-6-chloro-5-(methylpropylamino)-2-pyrazinecarboxamide;5-(N-Methyl-N-propyl)amiloride;MPA

Description

5-(N-methyl-N-propyl)amiloride is a member of the class of pyrazines that is amiloride in which the primary amino group adjacent to the chloro substiuent has been substituted by a methyl group and a propyl group. It has a role as a sodium channel blocker. It is a member of pyrazines, a member of guanidines, an organochlorine compound, a tertiary amino compound and a primary amino compound. It derives from an amiloride.

3-Amino-N-(aminoiminomethyl)-6-chloro-5-(methylpropylamino)-2-pyrazinecarboxamide Basic Attributes

285.736

285.73

Characteristics

137

1

214-215 °C

Drug Information

5-(N-methyl-N-propyl)amiloride

Computed Properties

Molecular Weight:285.73
XLogP3:1
Hydrogen Bond Donor Count:3
Hydrogen Bond Acceptor Count:5
Rotatable Bond Count:4
Exact Mass:285.1104859
Monoisotopic Mass:285.1104859
Topological Polar Surface Area:137
Heavy Atom Count:19
Complexity:347
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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