Product
Supplier
Encyclopedia
Inquiry
Home > Encyclopedia > Carvedilol phosphate

Carvedilol phosphate

pharmaceutical raw materials
Carvedilol phosphate structure

Carvedilol phosphate 

structure
  • CAS No:

    610309-89-2

  • Formula:

    C24H26N2O4.H3O4P.1/2H2O

  • Chemical Name:

    Carvedilol phosphate

  • Synonyms:

    2-Propanol,1-(9H-carbazol-4-yloxy)-3-[[2-(2-methoxyphenoxy)ethyl]amino]-,phosphate,hydrate (2:2:1);2-Propanol,1-(9H-carbazol-4-yloxy)-3-[[2-(2-methoxyphenoxy)ethyl]amino]-,phosphate (salt),hydrate (2:2:1);Carvedilol phosphate;SKF 105517D;Carvedilol phosphate hemihydrate;Carvedilol dihydrogen phosphate hemihydrate;Coreg CR

Description

Carvedilol is a non-selective beta blocker/alpha-1 blocker with an IC50 of 3.8 μM for inhibition of LDL oxidation.IC50 Value: 3.8 μM ( inhibition of LDL oxidation)Target: beta Adrenergic ReceptorCarvedilol is a nonselective-blocking agent and is used in the treatment of hypertension and angina pectoris. As a third-generation β-adrenergic blocker (β-blocker), Carvedilol is able to reverse cardiac structural remodeling. Recentresults demonstrated that the effect caused by Carvedilol on car

Carvedilol phosphate Basic Attributes

513.48

1026.34287

Characteristics

172.54000

3.13600

655.2ºC at 760 mmHg

350.1ºC

Safety Information

|Warning|H317 (100%): May cause an allergic skin reaction [Warning Sensitization, Skin]|P261, P272, P273, P280, P302+P352, P321, P333+P313, P363, P391, and P501|Aggregated GHS information provided by 2 companies from 1 notifications to the ECHA C&L Inventory. Each notification may be associated with multiple companies.

Carvedilol phosphate Use and Manufacturing

Uses

Treatment of congestive heart failure, left ventricular dysfunction following myocardial infarction, and management of hypertension.

Human Drugs -> FDA Approved Drug Products with Therapeutic Equivalence Evaluations (Orange Book) -> Active Ingredients

Computed Properties

Molecular Weight:1027.0
Hydrogen Bond Donor Count:13
Hydrogen Bond Acceptor Count:19
Rotatable Bond Count:20
Exact Mass:1026.34287045
Monoisotopic Mass:1026.34287045
Topological Polar Surface Area:308
Heavy Atom Count:71
Complexity:557
Undefined Atom Stereocenter Count:2
Covalently-Bonded Unit Count:5
Compound Is Canonicalized:Yes

Scan the QR Code to Share

Feedback & Suggestions
Send Message

Thank you for your feedback. If you require further assistance, please contact us by email at info@echemi.com or call us at +86-532-55729510.