Apixaban
19 Inquiries
503612-47-3
99%
2026-08-20
Coenzymes,Inhibito,Enzymes,Zymogens,Substrates,Native Microorganism Creatine Amidinohydrolase
-
Product Description
-
Seller Information
-
Inquiry History
-
Description
ProductName Apixaban Cat No CEI-0241 Description As a highly selective, reversible inhibitor, apixaban can inhibit Factor Xa with Ki of 0.08 nM and 0.17 nM in human and rabbit, respectively. CAS No 503612-47-3 Molecular Weight 459.5 Purity >99% Storage 2 years at -20 centigrade Targets Factor Xa Molecular Formula C25H25N5O4 Chemical Name 1-(4-methoxyphenyl)-7-oxo-6-(4-(2-oxopiperidin-1-yl)phenyl)-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxamide Solubility DSMO 18 mg/mL Water In vitro Apixaban exhibits a high degree of potency, selectivity, and efficacy on Factor Xa with Ki of 0.08 nM and 0.17 nM for Human Factor Xa and Rabbit Factor Xa. And Apixaban shows the highest potency in human and rabbit plasma. In vivo In the arteriovenous-shunt thrombosis (AVST), venous thrombosis (VT) and electrically mediated carotid arterial thrombosis (ECAT) rabbit models, Apixaban produces dose-dependent antithrombotic effects with EC50 of 270 nM, 110 nM and 70 nM. category Inhibitors(c1514) cas_num 503612-47-3 Basic Info-
Product Name:
Apixaban
Other Name:1H-Pyrazolo[3,4-c]pyridine-3-carboxamide,4,5,6,7-tetrahydro-1-(4-methoxyphenyl)-7-oxo-6-[4-(2-oxo-1-piperidinyl)phenyl]-;4,5,6,7-Tetrahydro-1-(4-methoxyphenyl)-7-oxo-6-[4-(2-oxo-1-piperidinyl)phenyl]-1H-pyrazolo[3,4-c]pyridine-3-carboxamide;1-(4-Methoxyphenyl)-7-oxo-6-[4-(2-oxopiperidin-1-yl)phenyl]-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylic acid amide;BMS 562247-01;Apixaban;Eliquis;1-(4-Methoxyphenyl)-7-oxo-6-[4-(2-oxopiperidin-1-yl)phenyl]-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxamide;1-(4-Methoxyphenyl)-7-oxo-6-[4-(2-oxopiperidin-1-yl)phenyl]-4,5-dihydropyrazolo[3,4-c]pyridine-3-carboxamide;1-(4-Methoxyphenyl)-7-oxo-6-[4-(2-oxopiperidin-1-yl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridine-3-carboxamide
CAS No.:503612-47-3
Molecular Formula:C25H25N5O4
InChIKeys:InChIKey=QNZCBYKSOIHPEH-UHFFFAOYSA-N
Molecular Weight:459.504
Exact Mass:459.50
Categories:
Characteristics-
PSA:
111
XLogP3:2.2
Density:1.42
Boiling Point:770.468ºC at 760 mmHg
Flash Point:419.8±32.9 °C
Refractive Index:1.705
Water Solubility:Aqueous solubility: 40-50 μg/ml in 0.9% saline solutionAqueous solubility across the physiological pH range is approximately 0.04 mg/L
Storage Conditions:Store at 20 deg C to 25 deg C (68 deg F-77 deg F); excursions permitted between 15 deg C and 30 deg C (59 deg F-86 deg F).
Vapor Pressure:4.29X10-18 mm Hg at 25 deg C (est)
Hazard IdentificationClassification of the substance or mixture
Specific target organ toxicity â repeated exposure, Category 1
GHS label elements, including precautionary statements
Pictogram(s) 
Signal word Danger
Hazard statement(s) H372 Causes damage to organs through prolonged or repeated exposure
Precautionary statement(s) Prevention P260 Do not breathe dust/fume/gas/mist/vapours/spray.
P264 Wash ... thoroughly after handling.
P270 Do not eat, drink or smoke when using this product.
Response P319 Get medical help if you feel unwell.
Storage none
Disposal P501 Dispose of contents/container to an appropriate treatment and disposal facility in accordance with applicable laws and regulations, and product characteristics at time of disposal.
Other hazards which do not result in classification
no data available
Handling and StoragePrecautions for safe handling
Handling in a well ventilated place. Wear suitable protective clothing. Avoid contact with skin and eyes. Avoid formation of dust and aerosols. Use non-sparking tools. Prevent fire caused by electrostatic discharge steam.
Conditions for safe storage, including any incompatibilities
Store the container tightly closed in a dry, cool and well-ventilated place. Store apart from foodstuff containers or incompatible materials.
-
-
Seller Information
-
Business Type:
Manufactory
-
Main Products:
Coenzymes,Inhibito,Enzymes,Zymogens,Substrates,Native Microorganism Creatine Amidinohydrolase
-
Location:
Shirley, New York 11967, USA
-
Payment Terms:
TT against copy of documents,D/P
-
Average lead Time:
15
-
Total Annual Revenue:
$1 million-$2.5 million
-
Year of Establishment:
2004
-
-
Inquiry History19 Inquiries
Country Product Purchase Quantity Date Posted 
India
Apixaban
50.00 KG May 29, 2025
India
Apixaban
20.00 KG May 27, 2025
India
Apixaban
20.00 KG May 27, 2025
India
Apixaban
40.00 KG May 27, 2025
India
Apixaban
10 G Jun 2, 2026
India
Apixaban
260.00 KG May 28, 2026
India
Apixaban
100 KG Dec 23, 2025
India
Apixaban
5 G Jul 4, 2025 
Italy
Apixaban
50.00 KG May 25, 2025
India
APIXABAN
1.00 KG Mar 25, 2025 
South Korea
Apixaban
100 KG Jan 25, 2024 
Brazil
Apixaban for wholesale
100 G Oct 25, 2023 
Bangladesh
Apixaban
300.00 KG May 30, 2025
India
Apixaban
100.00 KG Nov 11, 2023
India
ISOPROPYL ALCOHOL
20.00 KG May 27, 2025
India
Methanol
50.00 KG May 28, 2025
India
Cyclopentane
40.00 KG May 28, 2025 
Belgium
Linagliptin API
200.00 KG Jun 5, 2025
Belgium
Silicon dioxide
100.00 KG Jun 5, 2025 Post an enquiry for this product