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High Quality Pure 98% HPLC APD-125 Nelotanserin Raw Powder CAS 839713-36-9

Name: High Quality Pure 98% HPLC APD-125 Nelotanserin Raw Powder CAS 839713-36-9
Brand: HORLDEN
SKU: pr2511051377
Price: 700 USD
Availability: InStock

TDS 2 Inquiries

Unit Price:

$700-800/G FOB

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CAS No.:

839713-36-9

Grade:

Pharmaceutical Grade

Content:

99%

Port:

Shanghai

Brand:

HORLDEN

Packaging:

1g/bottle

Sample Available:

Yes

Price valid (until):

2026-11-08

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Xi'an Horlden Bio-Tech Co., Ltd

Company Type:

Trader

Location:

China

Payment Terms:

100% TT in advance

Average Lead Time:

7 days

Qualification:

Main Products:

Chemical,Intermediate,5-amino-1mq,SLU-PP332,Tirzepatide,Peptide

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Inquiry History

Description

Product Name	Nelotanserin
CAS NO.	839713-36-9
Purity	99%
Molecular formula	C18H15BrF2N4O2
MOQ	1 g

1-[3-(4-brom-1-methyl-1H-pyrazol-5-yl)-4-methoxypheyl]-3-(2,4-difluoropenyl)urea is a potent and complete inverse agonist of 5-HT2A, a moderately potent partial inverse agonist of 5-HT2C, and a weak inverse agonist of 5-HT2B, with IC50 values of 1.7, 79, and 791 nM, respectively.

You can ask us for quotation and product information via Email, Phone, WhatsApp and other channels.

Email: rock@horlden.com
WhatsApp/ Signal: +86 18829283179

1.What's your payment terms?

Standard terms: T/T in advance. Also L/C at sight is acceptable for large amount.

2.What's your shipping time?

We have bulk in stock, which means we can ship it to you immediately.

3.How do you ensure the quality of your products?

Strict QC with 6 steps testing from raw material purchase to finished product.

4.How do you ship the order normally?

For large qty order,ship the goods by sea. For small qty order, by air or express. We supply optional express for you, including DHL, FEDEX,UPS,TXT,EMS,and so on.

5.What's your loading port?

Usually Beijing, Shanghai, Qingdao, Tianjin, Guangzhou

ECHEMI Editorial Reference

Nelotanserin is a potent 5-HT2A inverse agonist, a moderately potent 5-HT2C partial inverse agonist and a weak 5-HT2B inverse agonist, with IC50s of 1.7, 79, 791 nM in IP accumulation assays, respectively.
Nelotanserin is a member of pyrazoles and a ring assembly.|Nelotanserin has been used in trials studying the treatment of Lewy Body Dementia, Visual Hallucinations, Dementia With Lewy Bodies, and REM Sleep Behavior Disorder. It is a highly selective antagonist at the 5-HT2A serotonin receptor. It increases non-REM sleep, the most restorative phase of the sleep cycle, without sacrificing REM or dream sleep. Nelotanserin works through a mechanism of action that is different from currently marketed drugs.

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Basic Info

Product Name:

N-[3-(4-Bromo-1-methyl-1H-pyrazol-5-yl)-4-methoxyphenyl]-N′-(2,4-difluorophenyl)urea

Other Name:

Urea,N-[3-(4-bromo-1-methyl-1H-pyrazol-5-yl)-4-methoxyphenyl]-N′-(2,4-difluorophenyl)-;N-[3-(4-Bromo-1-methyl-1H-pyrazol-5-yl)-4-methoxyphenyl]-N′-(2,4-difluorophenyl)urea;1-[3-(4-Bromo-2-methyl-2H-pyrazol-3-yl)-4-methoxyphenyl]-3-(2,4-difluorophenyl)urea;1-(2,4-Difluorophenyl)-3-[4-methoxy-3-(4-bromo-1-methyl-1H-pyrazol-5-yl)phenyl]urea;APD 125;Nelotanserin;1-[3-(4-Bromo-1-methyl-1H-pyrazol-5-yl)-4-methoxyphenyl]-3-(2,4-difluorophenyl)urea;1-[3-(4-Bromo-2-methylpyrazol-3-yl)-4-methoxyphenyl]-3-(2,4-difluorophenyl)urea

CAS No.:

839713-36-9

Molecular Formula:

C18H15BrF2N4O2

InChIKeys:

InChIKey=COSPVUFTLGQDQL-UHFFFAOYSA-N

Molecular Weight:

437.24

Exact Mass:

437.24

UNII:

4ZA73QEW2P

DSSTox ID:

DTXSID40232868

Categories:

Inhibitor Drugs

Characteristics

PSA:

68.2

XLogP3:

3.3

Density:

1.55 g/cm3

Boiling Point:

425.886°C at 760 mmHg

Flash Point:

211.369ºC

See More N-[3-(4-Bromo-1-methyl-1H-pyrazol-5-yl)-4-methoxyphenyl]-N′-(2,4-difluorophenyl)urea Properties 

Hazard Identification

Classification of the substance or mixture

no data available

GHS label elements, including precautionary statements

Precautionary statement(s)
Pictogram(s)	no data available
Signal word	no data available
Hazard statement(s)	no data available
Prevention	no data available
Response	no data available
Storage	no data available
Disposal	no data available

Other hazards which do not result in classification

no data available

Handling and Storage

Precautions for safe handling

Handling in a well ventilated place. Wear suitable protective clothing. Avoid contact with skin and eyes. Avoid formation of dust and aerosols. Use non-sparking tools. Prevent fire caused by electrostatic discharge steam.

Conditions for safe storage, including any incompatibilities

Store the container tightly closed in a dry, cool and well-ventilated place. Store apart from foodstuff containers or incompatible materials.

See More N-[3-(4-Bromo-1-methyl-1H-pyrazol-5-yl)-4-methoxyphenyl]-N′-(2,4-difluorophenyl)urea Safety Data Sheet 

Seller Information

Business Type:
Trader

Main Products:
Chemical,Intermediate,5-amino-1mq,SLU-PP332,Tirzepatide,Peptide

Location:
9th Floor, Room 923, Building 3, Shiyuan Daguan, Xingtai 1st Street, Chanba Ecological District, Xi'an City, Shaanxi Province

Payment Terms:
100% TT in advance

Average lead Time:
7 days

Total Annual Revenue:
$2.5 million-$5 million

Total Employees:
11-50

Year of Establishment:
2015

Xi'an Horlden Bio-Tech Co., Ltd is committed to promoting health application products such as chemical daily necessities, APIs, pharmaceutical intermediates and Cosmetic raw materials.

We have established friendly business relationships with hundreds of customers from over 50 countries and regions. Our team is committed to providing customers with the highest quality products at reasonable prices and satisfactory service. For many years, our company has won the trust and favor of our customers with high-quality products, first-class services, and competitive prices.

We will create the highest quality and most stable supply channel for customers, adhering to the spirit of serving customers, relying on strong funds and good cooperation reputation in the industry, to provide customers with higher quality products and services. At the same time, we are willing to strengthen exchanges and sincere cooperation with domestic and foreign merchants to create a better future together. It is your best supplier.

Welcome to Xi'an Horlden Bio-Tech Co., Ltd!

Inquiry History

2 Inquiries

Country	Product	Purchase Quantity	Date Posted
Netherlands	Nelotanserin	100 G	Nov 4, 2025
Spain	Nelotanserin	25 G	Apr 7, 2025

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Product Name	Grade / Content	Price	Supplier Name	Details
Nelotanserin	/99.00		HANGZHOU LEAP CHEM CO., LTD.	Inquiry

High Quality Pure 98% HPLC APD-125 Nelotanserin Raw Powder CAS 839713-36-9

Product Details

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