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Home > Encyclopedia > 3-Chloro-2-fluoropyridine-4-boronic acid

3-Chloro-2-fluoropyridine-4-boronic acid

3-Chloro-2-fluoropyridine-4-boronic acid structure

3-Chloro-2-fluoropyridine-4-boronic acid 

structure
  • CAS No:

    1217500-55-4

  • Formula:

    C5H4BClFNO2

  • Chemical Name:

    3-Chloro-2-fluoropyridine-4-boronic acid

  • Synonyms:

    3-Chloro-2-fluoropyridine-4-boronic acid;(3-Chloro-2-fluoropyridin-4-yl)boronic acid;Boronic acid, B-(3-chloro-2-fluoro-4-pyridinyl)-;MFCD09037477;3-Chloro-2-fluoropyridine-4-boronicacid;3-chloro-2-fluoropyridin-4-ylboronic acid;ACMC-209af7;CHEMBL3236589;CTK4B2629;KS-00000QEV

  • Categories:

    Pharmaceutical Intermediates  >  Heterocyclic Compound

3-Chloro-2-fluoropyridine-4-boronic acid Basic Attributes

175.3531632

175.00100

DTXSID50660294

Characteristics

53.4

1.51±0.1 g/cm3(Predicted)

126-130°C

349.6±52.0 °C(Predicted)

3-Chloro-2-fluoropyridine-4-boronic acid Use and Manufacturing

To a mixture of degassed 1 , 4-dioxane (2.8 mL) and water (0.64 mL) in a microwave vial was added [1 , 1 '-bis(diphenylphosphino)ferrocene]dichloropalladium(ll) complex with dichloromethane (0.0053 g, 0.0064 mmol), followed by the title compound from Preparative Example C (0.07 g, 0.127 mmol),

Computed Properties

Molecular Weight:175.35
Hydrogen Bond Donor Count:2
Hydrogen Bond Acceptor Count:4
Rotatable Bond Count:1
Exact Mass:175.0007644
Monoisotopic Mass:175.0007644
Topological Polar Surface Area:53.4
Heavy Atom Count:11
Complexity:140
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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