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Home > Encyclopedia > 1-O-Acetylbritannilactone

1-O-Acetylbritannilactone

1-O-Acetylbritannilactone structure

1-O-Acetylbritannilactone 

structure
  • CAS No:

    33627-41-7

  • Formula:

    C17H24O5

  • Chemical Name:

    1-O-Acetylbritannilactone

  • Synonyms:

    2(3H)-Benzofuranone,5-[(1S)-4-(acetyloxy)-1-methylbutyl]-3a,4,7,7a-tetrahydro-4-hydroxy-6-methyl-3-methylene-,(3aS,4S,7aR)-;2(3H)-Benzofuranone,5-[4-(acetyloxy)-1-methylbutyl]-3a,4,7,7a-tetrahydro-4-hydroxy-6-methyl-3-methylene-,[3aS-[3aα,4α,5(R*),7aα]]-;(3aS,4S,7aR)-5-[(1S)-4-(Acetyloxy)-1-methylbutyl]-3a,4,7,7a-tetrahydro-4-hydroxy-6-methyl-3-methylene-2(3H)-benzofuranone;Inulicin;1-O-Acetylbritannilactone;1-O-Acetylbritannilatone;Britannilactone 1-O-acetate;1-Acetoxy-6α-hydroxyeriolanolide;681457-46-5;744203-09-6

  • Categories:

    Biochemical Engineering  >  Chinese Herbs

Description

1-O-Acetylbritannilactone is an active compound isolated from Inula Britannica L. 1-O-Acetylbritannilactone inhibits VEGF-mediated activation of Src and FAK. 1-O-Acetylbritannilactone inhibits LPS-induced PGE2 production and COX-2 expression, and NF-κB activation and translocation.

1-O-Acetylbritannilactone Basic Attributes

308.372

308.37

Characteristics

72.83000

2.12

1.2±0.1 g/cm3

124.0-126.1 °C

483.1±45.0 °C at 760 mmHg

173.1±22.2 °C

1.521

Computed Properties

Molecular Weight:308.4
XLogP3:1.3
Hydrogen Bond Donor Count:1
Hydrogen Bond Acceptor Count:5
Rotatable Bond Count:6
Exact Mass:308.16237386
Monoisotopic Mass:308.16237386
Topological Polar Surface Area:72.8
Heavy Atom Count:22
Complexity:519
Undefined Atom Stereocenter Count:4
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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