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Home > Encyclopedia > 3,4-Dihydro-4-hydroxy-2(1H)-isoquinolinecarboximidamide

3,4-Dihydro-4-hydroxy-2(1H)-isoquinolinecarboximidamide

3,4-Dihydro-4-hydroxy-2(1H)-isoquinolinecarboximidamide structure

3,4-Dihydro-4-hydroxy-2(1H)-isoquinolinecarboximidamide 

structure
  • CAS No:

    59333-79-8

  • Formula:

    C10H13N3O

  • Chemical Name:

    3,4-Dihydro-4-hydroxy-2(1H)-isoquinolinecarboximidamide

  • Synonyms:

    2(1H)-Isoquinolinecarboximidamide,3,4-dihydro-4-hydroxy-;3,4-Dihydro-4-hydroxy-2(1H)-isoquinolinecarboximidamide;Ro 03-7594;4-Hydroxydebrisoquin;Ro 3-7594/001;(±)-4-Hydroxydebrisoquine;114673-70-0

  • Categories:

    Chemical Reagents  >  Organic Reagents

Description

ChEBI: An isoquinoline that is 3,4-dihydroisoquinoline bearing amidino and hydroxy substituent at positions 2 and 4 respectively.


Solid


4-hydroxydebrisoquin is an isoquinoline that is 3,4-dihydroisoquinoline bearing amidino and hydroxy substituent at positions 2 and 4 respectively. It has a role as a metabolite. It is a carboxamidine, a member of isoquinolines and a secondary alcohol.

3,4-Dihydro-4-hydroxy-2(1H)-isoquinolinecarboximidamide Basic Attributes

191.23

191.23

2933499090

Characteristics

73.3

1.16700

1.38g/cm3

374.2ºC at 760 mmHg

180.1ºC

1.679

Drug Information

4-Hydroxydebrisoquine is a known human metabolite of debrisoquine.

4-hydroxydebrisoquin

Computed Properties

Molecular Weight:191.23
XLogP3:-0.3
Hydrogen Bond Donor Count:3
Hydrogen Bond Acceptor Count:2
Rotatable Bond Count:1
Exact Mass:191.105862047
Monoisotopic Mass:191.105862047
Topological Polar Surface Area:73.3
Heavy Atom Count:14
Complexity:231
Undefined Atom Stereocenter Count:1
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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