Product
Supplier
Encyclopedia
Inquiry
Home > Encyclopedia > (αR,βS)-α-(4-Hydroxyphenyl)-β-methyl-4-(phenylmethyl)-1-piperidinepropanol

(αR,βS)-α-(4-Hydroxyphenyl)-β-methyl-4-(phenylmethyl)-1-piperidinepropanol

(αR,βS)-α-(4-Hydroxyphenyl)-β-methyl-4-(phenylmethyl)-1-piperidinepropanol structure

(αR,βS)-α-(4-Hydroxyphenyl)-β-methyl-4-(phenylmethyl)-1-piperidinepropanol 

structure
  • CAS No:

    169274-78-6

  • Formula:

    C22H29NO2

  • Chemical Name:

    (αR,βS)-α-(4-Hydroxyphenyl)-β-methyl-4-(phenylmethyl)-1-piperidinepropanol

  • Synonyms:

    1-Piperidinepropanol,α-(4-hydroxyphenyl)-β-methyl-4-(phenylmethyl)-,(αR,βS)-;1-Piperidinepropanol,α-(4-hydroxyphenyl)-β-methyl-4-(phenylmethyl)-,[R-(R*,S*)]-;(αR,βS)-α-(4-Hydroxyphenyl)-β-methyl-4-(phenylmethyl)-1-piperidinepropanol;Ro 25-6981

Description

4-[(1R,2S)-1-hydroxy-2-methyl-3-[4-(phenylmethyl)-1-piperidinyl]propyl]phenol is a member of piperidines.

(αR,βS)-α-(4-Hydroxyphenyl)-β-methyl-4-(phenylmethyl)-1-piperidinepropanol Basic Attributes

455.54

339.47

DTXSID20849493

Characteristics

43.7 Ų

3.66610

1.116±0.06 g/cm3(Predicted)

512.4±45.0 °C(Predicted)

379.4ºC

1.587

Desiccate at RT

2.52E-11mmHg at 25°C

Drug Information

alpha-(4-hydroxyphenyl)-beta-methyl--4-(phenylmethyl)-1-piperidine propanol

(αR,βS)-α-(4-Hydroxyphenyl)-β-methyl-4-(phenylmethyl)-1-piperidinepropanol Use and Manufacturing

Potent and selective activity-dependent blocker of NMDA receptors containing the NR2B subunit. IC 50 values are 0.009 and 52 μ M for cloned receptor subunit combinations NR1C/NR2B and NR1C/NR2A respectively. Displays neuroprotectant effects in vivo and in vitro .

Computed Properties

Molecular Weight:339.5
XLogP3:4.2
Hydrogen Bond Donor Count:2
Hydrogen Bond Acceptor Count:3
Rotatable Bond Count:6
Exact Mass:339.219829168
Monoisotopic Mass:339.219829168
Topological Polar Surface Area:43.7
Heavy Atom Count:25
Complexity:366
Defined Atom Stereocenter Count:2
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

Scan the QR Code to Share

Feedback & Suggestions
Send Message

Thank you for your feedback. If you require further assistance, please contact us by email at info@echemi.com or call us at +86-532-55729510.