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Home > Encyclopedia > BMS-740808

BMS-740808

BMS-740808 structure

BMS-740808 

structure
  • CAS No:

    280118-23-2

  • Formula:

    C31H27F3N6O3

  • Chemical Name:

    BMS-740808

  • Synonyms:

    1-(3-aminobenzisoxazol-5"-yl)-3-trifluoromethyl-6-(2"-(3-hydroxy-N-pyrrolidinyl)methyl-(1,1")-biphen-4-yl)-1,4,5,6-tetrahydropyrazolo-(3,4-c)-pyridin-7-one;BMS 740808;BMS-740808;BMS740808;UNII-LDD74E663F;LDD74E663F;1-(3-AMINO-1,2-BENZISOXAZOL-5-YL)-6-(2"-{[(3R)-3-HYDROXYPYRROLIDIN-1-YL]METHYL}BIPHENYL-4-YL)-3-(TRIFLUOROMETHYL)-1,4,5,6-TETRAHYDRO-7H-PYRAZOLO[3,4-C]PYRIDIN-7-ONE

BMS-740808 Basic Attributes

588.591

588.21

LDD74E663F

DTXSID40182293

Characteristics

114

4.6

1.52

Drug Information

Endogenous factors and drugs that inhibit or block the activity of FACTOR XA. (See all compounds classified as Factor Xa Inhibitors.)

1-(3-aminobenzisoxazol-5'-yl)-3-trifluoromethyl-6-(2'-(3-hydroxy-N-pyrrolidinyl)methyl-(1,1')-biphen-4-yl)-1,4,5,6-tetrahydropyrazolo-(3,4-c)-pyridin-7-one

Computed Properties

Molecular Weight:588.6
XLogP3:4.6
Hydrogen Bond Donor Count:2
Hydrogen Bond Acceptor Count:10
Rotatable Bond Count:5
Exact Mass:588.20967323
Monoisotopic Mass:588.20967323
Topological Polar Surface Area:114
Heavy Atom Count:43
Complexity:998
Defined Atom Stereocenter Count:1
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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