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Tecastemizole

Tecastemizole structure

Tecastemizole 

structure
  • CAS No:

    75970-99-9

  • Formula:

    C19H21FN4

  • Chemical Name:

    Tecastemizole

  • Synonyms:

    1H-Benzimidazol-2-amine,1-[(4-fluorophenyl)methyl]-N-4-piperidinyl-;1-[(4-Fluorophenyl)methyl]-N-4-piperidinyl-1H-benzimidazol-2-amine;1-(4-Fluorobenzyl)-2-(4-piperidylamino)benzimidazole;1-(4-Fluorophenylmethyl)-2-(4-piperidylamino)benzimidazole;Norastemizole;T 1348;Soltara;Tecastemizole

Tecastemizole Basic Attributes

324.39500

324.40

W5DCO14M05

DTXSID30226877

Characteristics

45.11000

3.13830

1.28g/cm3

290.2 °C

519.8ºC

268.2ºC

1.658

Drug Information

Investigated for use/treatment in allergic rhinitis.

Norastemizole is a known human metabolite of astemizole.

1-((4-flurophenyl)methyl)-N-4-piperidinyl-1H-benzimidazol-2-amine

Computed Properties

Molecular Weight:324.4
XLogP3:3.6
Hydrogen Bond Donor Count:2
Hydrogen Bond Acceptor Count:4
Rotatable Bond Count:4
Exact Mass:324.17502485
Monoisotopic Mass:324.17502485
Topological Polar Surface Area:41.9
Heavy Atom Count:24
Complexity:393
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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