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Iododoxorubicin

Iododoxorubicin structure

Iododoxorubicin 

structure
  • CAS No:

    83997-75-5

  • Formula:

    C27H28INO10

  • Chemical Name:

    Iododoxorubicin

  • Synonyms:

    5,12-Naphthacenedione,10-[[(2R,4S,5S,6S)-4-aminotetrahydro-5-iodo-6-methyl-2H-pyran-2-yl]oxy]-7,8,9,10-tetrahydro-6,8,11-trihydroxy-8-(2-hydroxyacetyl)-1-methoxy-,(8S,10S)-;5,12-Naphthacenedione,10-[[(2R,4S,5S,6S)-4-aminotetrahydro-5-iodo-6-methyl-2H-pyran-2-yl]oxy]-7,8,9,10-tetrahydro-6,8,11-trihydroxy-8-(hydroxyacetyl)-1-methoxy-,(8S,10S)-;(8S,10S)-10-[[(2R,4S,5S,6S)-4-Aminotetrahydro-5-iodo-6-methyl-2H-pyran-2-yl]oxy]-7,8,9,10-tetrahydro-6,8,11-trihydroxy-8-(2-hydroxyacetyl)-1-methoxy-5,12-naphthacenedione;4′-Deoxy-4′-iododoxorubicin;4′-Deoxy-4′-iodoadriamycin;4′-Iodo-4′-deoxydoxorubicin;FCE 21954;Iododoxorubicin;WP 154;119485-06-2;144120-06-9

  • Categories:

    Biochemical Engineering  >  Saccharides

Description

4'-deoxy-4'-iododoxorubicin is an organoiodine compound, a primary alpha-hydroxy ketone and a tertiary alpha-hydroxy ketone. It derives from a doxorubicin. It is a conjugate acid of a 4'-deoxy-4'-iododoxorubicinium.|4'-Iodo-4'-Deoxydoxorubicin is an iodinated doxorubicin analogue with antiamyloid activity. 4'-Iodo-4'-deoxydoxorubicin (IDOX) binds with high affinity to five types of natural amyloid fibrils including immunoglobulin light chains, amyloid A, transthyretin (methionine-30 variant), beta-protein (Alzheimer), and beta2-microglobulin. This agent may inhibit fibril growth, increasing the solubility of amyloid tissue deposits and facilitating their clearance. IDOX has also been shown to insulin amyloid fibrillogenesis in vitro.

Iododoxorubicin Basic Attributes

653.41600

653.42

65JH75I9JX

C971

Characteristics

185.84000

2.83440

1.81g/cm3

813.2ºC at 760 mmHg

445.6ºC

1.727

Drug Information

4'-deoxy-4'-IDX

Computed Properties

Molecular Weight:653.4
XLogP3:2.9
Hydrogen Bond Donor Count:5
Hydrogen Bond Acceptor Count:11
Rotatable Bond Count:5
Exact Mass:653.07579
Monoisotopic Mass:653.07579
Topological Polar Surface Area:186
Heavy Atom Count:39
Complexity:982
Defined Atom Stereocenter Count:6
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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