Product
Supplier
Encyclopedia
Inquiry
Home > Encyclopedia > Amrubicin hydrochloride

Amrubicin hydrochloride

pharmaceutical raw materials
Amrubicin hydrochloride structure

Amrubicin hydrochloride 

structure
  • CAS No:

    110311-30-3

  • Formula:

    C25H25NO9.ClH

  • Chemical Name:

    Amrubicin hydrochloride

  • Synonyms:

    5,12-Naphthacenedione,9-acetyl-9-amino-7-[(2-deoxy-β-D-erythro-pentopyranosyl)oxy]-7,8,9,10-tetrahydro-6,11-dihydroxy-,hydrochloride (1:1),(7S,9S)-;5,12-Naphthacenedione,9-acetyl-9-amino-7-[(2-deoxy-β-D-erythro-pentopyranosyl)oxy]-7,8,9,10-tetrahydro-6,11-dihydroxy-,hydrochloride,(7S-cis)-;5,12-Naphthacenedione,9-acetyl-9-amino-7-[(2-deoxy-β-D-erythro-pentopyranosyl)oxy]-7,8,9,10-tetrahydro-6,11-dihydroxy-,hydrochloride,(7S,9S)-;SM 5887;Amrubicin hydrochloride;Calsed

Description

Amrubicin Hydrochloride is the hydrochloride salt of a third-generation synthetic 9-amino-anthracycline with antineoplastic activity. Amrubicin intercalates into DNA and inhibits the activity of topoisomerase II, resulting in inhibition of DNA replication, and RNA and protein synthesis, followed by cell growth inhibition and cell death. This agent has demonstrated a higher level of anti-tumor activity than conventional anthracycline drugs without exhibiting any indication of the cumulative cardiac toxicity common to this class of compounds.

Amrubicin hydrochloride Basic Attributes

519.9 g/mol

519.1296091 g/mol

EUL6MP8FZW

C47948

Characteristics

177 Ų

Drug Information

Substances that inhibit or prevent the proliferation of NEOPLASMS. (See all compounds classified as Antineoplastic Agents.)

(+)-(7S,9S)-9-acetyl-9-amino-7-((2-deoxy-beta-d-erythro-pentopyranosyl)oxy)-6,11-dihydroxy-7,8,9,10-tetrahydrotetracene-5,12-dione hydrochloride

Amrubicin hydrochloride Use and Manufacturing

Human drugs -> Rare disease (orphan)

Computed Properties

Molecular Weight:519.9
Hydrogen Bond Donor Count:6
Hydrogen Bond Acceptor Count:10
Rotatable Bond Count:3
Exact Mass:519.1296091
Monoisotopic Mass:519.1296091
Topological Polar Surface Area:177
Heavy Atom Count:36
Complexity:881
Defined Atom Stereocenter Count:5
Covalently-Bonded Unit Count:2
Compound Is Canonicalized:Yes

Scan the QR Code to Share

Feedback & Suggestions
Send Message

Thank you for your feedback. If you require further assistance, please contact us by email at info@echemi.com or call us at +86-532-55729510.