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Scoulerine

Scoulerine structure

Scoulerine 

structure
  • CAS No:

    6451-73-6

  • Formula:

    C19H21NO4

  • Chemical Name:

    Scoulerine

  • Synonyms:

    6H-Dibenzo[a,g]quinolizine-2,9-diol,5,8,13,13a-tetrahydro-3,10-dimethoxy-,(13aS)-;13aα-Berbine-2,9-diol,3,10-dimethoxy-;6H-Dibenzo[a,g]quinolizine-2,9-diol,5,8,13,13a-tetrahydro-3,10-dimethoxy-,(S)-;Scoulerine;(13aS)-5,8,13,13a-Tetrahydro-3,10-dimethoxy-6H-dibenzo[a,g]quinolizine-2,9-diol;(-)-Scoulerine;Scoulerine,(-)-;Alkaloid HF 1,from Hunnemanniafumariaefolia;l-Scoulerine;(S)-(-)-Scoulerine;Scoulerin;(S)-Scoulerine;(13AS)-3,10-dimethoxy-6,8,13,13a-tetrahydro-5H-isoquinolino[2,1-b]isoquinoline-2,9-diol

  • Categories:

    Natural Products  >  Alkaloids

Description

Off-White to Pale Pink Solid


(S)-scoulerine is a berberine alkaloid isolated from Corydalis saxicola. It has a role as an EC 5.99.1.2 (DNA topoisomerase) inhibitor and a plant metabolite. It is an organic heterotetracyclic compound and a berberine alkaloid.

Scoulerine Basic Attributes

327.37

327.37

Characteristics

62.2

2.16

1.4±0.1 g/cm3

195-196 °C

503.3±50.0 °C at 760 mmHg

258.2±30.1 °C

1.680

Drug Information

aequaline

Scoulerine Use and Manufacturing

(S)-Scoulerine is an alkaloid found in the opium poppy. (S)-Scoulerine acts as an antagonist at the α2-adrenoceptor, α1D-adrenoceptor and 5-HT receptor.

Computed Properties

Molecular Weight:327.4
XLogP3:2.6
Hydrogen Bond Donor Count:2
Hydrogen Bond Acceptor Count:5
Rotatable Bond Count:2
Exact Mass:327.14705815
Monoisotopic Mass:327.14705815
Topological Polar Surface Area:62.2
Heavy Atom Count:24
Complexity:447
Defined Atom Stereocenter Count:1
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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