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Quinisocaine

Quinisocaine structure

Quinisocaine 

structure
  • CAS No:

    86-80-6

  • Formula:

    C17H24N2O

  • Chemical Name:

    Quinisocaine

  • Synonyms:

    Ethanamine,2-[(3-butyl-1-isoquinolinyl)oxy]-N,N-dimethyl-;Isoquinoline,3-butyl-1-[2-(dimethylamino)ethoxy]-;2-[(3-Butyl-1-isoquinolinyl)oxy]-N,N-dimethylethanamine;Dimethisoquin;1-(β-Dimethylaminoethoxy)-3-n-butylisoquinoline;Pruralgan;Quinisocaine;Chinisocain;Histaderme;Prulantex;Quinisocain;Quinoleine;Kinisocaine;[2-[(3-Butylisoquinolin-1-yl)oxy]ethyl]dimethylamine

Description

2-[(3-butyl-1-isoquinolinyl)oxy]-N,N-dimethylethanamine is a member of isoquinolines.

Quinisocaine Basic Attributes

272.38500

272.39

201-700-0

772EN3BH6I

39695

DTXSID8048525

D - Dermatologicals

Characteristics

25.36000

3.51780

1.034g/cm3

146 °C

155-157 °C @ Press: 3 Torr

188.6ºC

1.561

Drug Information

Drugs that block nerve conduction when applied locally to nerve tissue in appropriate concentrations. They act on any part of the nervous system and on every type of nerve fiber. In contact with a nerve trunk, these anesthetics can cause both sensory and motor paralysis in the innervated area. Their action is completely reversible. (From Gilman AG, et. al., Goodman and Gilman's The Pharmacological Basis of Therapeutics, 8th ed) Nearly all local anesthetics act by reducing the tendency of voltage-dependent sodium channels to activate. (See all compounds classified as Anesthetics, Local.)

3-butyl-1-(2-dimethylaminoethoxy)isoquinoline

Quinisocaine Use and Manufacturing

Pharmaceuticals

Computed Properties

Molecular Weight:272.4
XLogP3:4.2
Hydrogen Bond Acceptor Count:3
Rotatable Bond Count:7
Exact Mass:272.188863393
Monoisotopic Mass:272.188863393
Topological Polar Surface Area:25.4
Heavy Atom Count:20
Complexity:270
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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