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Oxabolone cipionate

Oxabolone cipionate structure

CAS No:
1254-35-9
Formula:
C26H38O4
Chemical Name:
Oxabolone cipionate
Synonyms:
Estr-4-en-3-one,17-(3-cyclopentyl-1-oxopropoxy)-4-hydroxy-,(17β)-;Estr-4-en-3-one,4,17β-dihydroxy-,17-cyclopentanepropionate;(17β)-17-(3-Cyclopentyl-1-oxopropoxy)-4-hydroxyestr-4-en-3-one;Cyclopentanepropionic acid,17-ester with 4,17β-dihydroxyestr-4-en-3-one;4-Hydroxy-19-nortestosterone 17-cyclopentylpropionate;4-Hydroxy-19-nortestosterone 17-cyclopentanepropionate;4-Hydroxy-19-nortestosterone cyclopentanepropionate;4-Hydroxy-19-nortestosterone-17-cyclopentapropionate;Oxabolone cipionate;Steranabol Long-Acting;FI 5852;Oxabolone 17-cyclopentanepropionate;Steranabol ritardo;NSC 522767
Categories:
Pharmaceutical Intermediates > Bulk Drug Intermediates

Description

Oxabolone cipionate is an organic molecular entity.|Oxabolone cipionate is the C17β cypionate ester and a prodrug of [DB01500]. A synthetic anabolic-androgenic (AAS) steroid, it is a derivative of 19-nortestosterone (nandrolone). It is considered as a performance enhancing drug thus is prohibited from use in sports.

Oxabolone cipionate Basic Attributes

Molecular Weight：

414.57800

Exact Mass：

414.58

EC Number：

215-011-8

UNII：

5RXY50Q01N

DSSTox ID：

DTXSID3046879

ATC Code：

A - Alimentary tract and metabolism

Characteristics

PSA：

63.60000

XLogP3：

5.89610

Density：

1.16g/cm3

Melting Point：

158-160 °C

Boiling Point：

560.7ºC at 760mmHg

Flash Point：

184.9ºC

Refractive Index：

1.561

Drug Information

Drug Indication：

Used as a performance enhancing drug illicitly in athletes.

Pharmacology：

Androgenic effects include enhanced secondary sexual characteristics.

Absorption：

The metabolites and unchanged form of oxabolone can be detected in the urine.|The elimination on the first day following intravenous injection of oxabolone cipionate is slow and reaches a rapid excretion phase with the maximum urinary level in the fifth day of administration.

Metabolism/Metabolites：

The prodrug oxabolone cipionate is converted to oxabolone. Oxabolone is then metabolized into 4-Hydroxyestr-4-en-3,17-dione (M2) which is the most abundant metabolite via oxidation of the 17-hydroxyl group. 4-Hydroxyestran-3,17-dione (M1) is formed by reduction of the A ring double bond along with the oxidation of the 17-hydroxyl group. Three isomeric compounds exist as another metabolite, as the 3α,4-dihydroxy-5α-estran-17-one, 3α,4-dihydroxy-5β-estran-17-one, and 3β,4-dihydroxy-5α-estran-17-one.

MeSH Entry Terms：

4,17beta-dihydroxy-estr-4-en-3-one 17-cyclopentylpropionate

Computed Properties

Molecular Weight:414.6
XLogP3:5.7
Hydrogen Bond Donor Count:1
Hydrogen Bond Acceptor Count:4
Rotatable Bond Count:5
Exact Mass:414.27700969
Monoisotopic Mass:414.27700969
Topological Polar Surface Area:63.6
Heavy Atom Count:30
Complexity:733
Defined Atom Stereocenter Count:6
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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Oxabolon cipionate 1254-35-9

Unit Price: $300-330 /KG FOB

CAS No.: 1254-35-9

Grade: Cosmetics Grade

Content: 99%

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