Sulpiride Injection
Function and Efficacy
This product belongs to the benzamide antipsychotic drug. Its characteristic action is to selectively block the dopamine (DA2) receptors of the mesolimbic system, with little effect on other neurotransmitter receptors, mild anticholinergic effect, and no obvious sedative and anti-excitement and agitation effects. This product also has strong antiemetic and gastric juice secretion inhibitory effects.
Ingredients
The main ingredient of this product is Sulpiride, and its chemical name is: N-[methyl-(1-ethyl-2-pyrrolidinyl)]-2-methoxy-5-(aminosulfonyl)-benzamide.
| Name | Description | Content | CAS NO. | Manufacturer |
|---|---|---|---|---|
| SulpirideIngredients |
This product belongs to the benzamide antipsychotic drug. Its characteristic action is to selectively block the dopamine (DA2) receptors of the mesolimbic system, with little effect on other neurotransmitter receptors, mild anticholinergic effect, and no obvious sedative and anti-excitement and agitation effects. This product also has strong antiemetic and gastric juice secretion inhibitory effects. More |
15676-16-1 | 12 |
Appearance
This product is a colorless clear liquid.
Indication
It has a good effect on apathy, withdrawal, stupor, depression, hallucination and delusion. It is suitable for simple schizophrenia, paranoid schizophrenia, tension type, and chronic schizophrenia. It has a certain effect on depression. It has no obvious sedative and anti-excitement effect. Other uses include anti-vomiting.
Usage and Dosage
For the treatment of schizophrenia, intramuscular injection: 100 mg once, twice a day. Intravenous drip: For patients with stupor and rebelliousness, 100-200 mg of this product can be diluted in 250-500 ml of glucose and sodium chloride injection and slowly dripped intravenously, once a day, and can be gradually increased to 300-600 mg per day, and the daily dose should not exceed 800 mg. The drip time should be no less than 4 hours.
Adverse Reactions
1 Common symptoms include insomnia, early awakening, headache, irritability, fatigue, loss of appetite, etc. Anticholinergic adverse reactions such as dry mouth, blurred vision, tachycardia, dysuria and constipation may occur. 2 Extrapyramidal reactions such as tremor, rigidity, drooling, bradykinesia, akathisia, and acute dystonia may occur when the dose is greater than 600 mg per day. 3 It often causes an increase in plasma prolactin concentration, and the possible related symptoms are: galactorrhea, gynecomastia, menstrual disorders, amenorrhea, and weight gain. 4 Electrocardiogram abnormalities and liver damage may occur. 5 A small number of patients may experience excitement, agitation, sleep disorders or increased blood pressure. 6
Precautions
It is contraindicated for patients with pheochromocytoma, hypertension, severe cardiovascular disease, severe liver disease, or those who are allergic to this product.
Drug Interactions
Except for clozapine, almost all antipsychotics and central nervous system depressants interact with it and should be treated with full attention.
Storage
Keep away from light and store in a sealed container.
Packaging Specification
2ml:0.1g
Manufacturer
Hunan Dongting Pharmaceutical Co., Ltd.
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Founded in:
1997-03-26 -
Address:
No. 16 Dongyan Road, Chenjiagang Community, Deshan Subdistrict Office, Changde Economic and Technological Development Zone, Hunan Province (No. 16 Dongyan Road, Deshan District, Changde City) -
Tax NO.:
914307001838043692 -
Registered Funds:
309.624852 million yuan -
Website:
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Email: