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High Purity 99% Sitagliptin Powder CAS 486460-32-6

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CAS No.:

486460-32-6

Content:

Packaging:

Foil Bag, Box, Drum

Sample Available:

Yes

Price valid (until):

2022-12-31

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Xian ZB Biotech Co.,Ltd

Company Type:

Manufactory

Location:

China

Payment Terms:

TT against copy of documents

Average Lead Time:

8 days

Qualification:

Main Products:

Herb Extracts,Cosmetic raw materails,API

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Product Details
Seller Information
Inquiry History

Description

Product Description

_{Prodcut name}	_Sitagliptin
_Synonyms	_{(3R)-3-Amino-1-[3-(trifluoromethyl)-5,6,7,8-tetrahydro-1,2,4-triazolo[4,3-a]pyrazin-7-yl]-4-(2,4,5-trifluorophenyl)butan-1-one}
_MOQ	_1G
_{CAS No.}	_486460-32-6
_Appearance	_{white powder}
_{Molecular Formula}	_C16H15F6N5O
_{Molecular Weight}	_407.32
_Assay	_99%
_Application	_{Pharma grade or research purpose}
_Packing	_{As per your request}
_Storage	_{Preserve in tight,light-resistant containers in a cool place}
_Remarks	_NA
_{Custom synthesis}	_Available
_{Supply Ability}	_500kg/month

_{Specification:}

_{I tems}	_{S tandards}	_{R esults}
_Appearance	_{White to off-white crystalline powder}	_Complies
_{I dentification}	_{By IR}	_Complies
	_{By HPLC}	_Complies
	_Phosphate	_Complies
_Solubility	_{Freely soluble in Water}	_Complies
_{Water Content(KF)}	_3.3%~3.7%	_3.49%
_{Residue on Ignition}	_{≤ 0.20%}	_0.06%
_{H eavy M etals}	_{≤ 20ppm}	_Complies
_{Chiral Impurity}	_{≤ 0.50%}	_ND
_{R elated S ubstances}	_{Any individual impurity: ≤0.10%}	_0.04%
	_{Total impurities: ≤0.50%}	_0.07%
_{Assay (HPLC basis on drying)}	_98.0%~102.0%	_99.88%
_{Reference Standard}	_{USP39 Standard}
_Conclusion	_{The product complie d to USP39 standard .}
_Storage	_{Preserve in tight,light-resistant containers in a cool place}

ECHEMI Editorial Reference

Sitagliptin is a potent inhibitor of DPP4 with IC50 of 19 nM in Caco-2 cell extracts.

Certificates

Basic Info

Product Name:

Sitagliptin

Other Name:

1-Butanone,3-amino-1-[5,6-dihydro-3-(trifluoromethyl)-1,2,4-triazolo[4,3-a]pyrazin-7(8H)-yl]-4-(2,4,5-trifluorophenyl)-,(3R)-;1,2,4-Triazolo[4,3-a]pyrazine,7-[(3R)-3-amino-1-oxo-4-(2,4,5-trifluorophenyl)butyl]-5,6,7,8-tetrahydro-3-(trifluoromethyl)-;(3R)-3-Amino-1-[5,6-dihydro-3-(trifluoromethyl)-1,2,4-triazolo[4,3-a]pyrazin-7(8H)-yl]-4-(2,4,5-trifluorophenyl)-1-butanone;(2R)-4-Oxo-4-[3-(trifluoromethyl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl]-1-(2,4,5-trifluorophenyl)butan-2-amine;Sitagliptin;3(R)-Amino-1-[3-(trifluoromethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-4-(2,4,5-trifluorophenyl)butan-1-one;7-[(3R)-3-Amino-1-oxo-4-(2,4,5-trifluorophenyl)butyl]-5,6,7,8-tetrahydro-3-(trifluoromethyl)-1,2,4-triazolo[4,3-a]pyrazine;(3R)-3-Amino-1-[3-(trifluoromethyl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-4-(2,4,5-trifluorophenyl)butan-1-one;(3R)-3-Amino-1-[3-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-4-(2,4,5-trifluorophenyl)butan-1-one;Xelevia;Tesavel;Ristaben

CAS No.:

486460-32-6

Molecular Formula:

C16H15F6N5O

InChIKeys:

InChIKey=MFFMDFFZMYYVKS-SECBINFHSA-N

Molecular Weight:

407.32

Exact Mass:

407.31

EC Number:

1308068-626-2

Categories:

Circulatory System Drugs

Characteristics

PSA:

XLogP3:

1.5

Appearance:

Solid

Density:

1.6±0.1 g/cm3

Melting Point:

114.1-115.7 °C

Boiling Point:

529.9±60.0 °C at 760 mmHg

Flash Point:

274.3±32.9 °C

Refractive Index:

1.590

Water Solubility:

3.40e-02 g/L

Storage Conditions:

Store at 20-25 deg C (68-77 deg F), excursions permitted to 15-30 deg C (59-86 deg F).

Vapor Pressure:

2.91X10-8 mm Hg at 25 deg C (est)

See More Sitagliptin Properties 

Hazard Identification

Classification of the substance or mixture

Acute toxicity - Category 4, Oral

Serious eye damage, Category 1

Specific target organ toxicity â repeated exposure, Category 2

GHS label elements, including precautionary statements

Precautionary statement(s)
Pictogram(s)
Signal word	Danger
Hazard statement(s)	H302 Harmful if swallowed H318 Causes serious eye damage H373 May cause damage to organs through prolonged or repeated exposure
Prevention	P264 Wash ... thoroughly after handling. P270 Do not eat, drink or smoke when using this product. P280 Wear protective gloves/protective clothing/eye protection/face protection/hearing protection/... P260 Do not breathe dust/fume/gas/mist/vapours/spray.
Response	P301+P317 IF SWALLOWED: Get medical help. P330 Rinse mouth. P305+P354+P338 IF IN EYES: Immediately rinse with water for several minutes. Remove contact lenses, if present and easy to do. Continue rinsing. P317 Get medical help. P319 Get medical help if you feel unwell.
Storage	none
Disposal	P501 Dispose of contents/container to an appropriate treatment and disposal facility in accordance with applicable laws and regulations, and product characteristics at time of disposal.

Other hazards which do not result in classification

no data available

Handling and Storage

Precautions for safe handling

Handling in a well ventilated place. Wear suitable protective clothing. Avoid contact with skin and eyes. Avoid formation of dust and aerosols. Use non-sparking tools. Prevent fire caused by electrostatic discharge steam.

Conditions for safe storage, including any incompatibilities

Store the container tightly closed in a dry, cool and well-ventilated place. Store apart from foodstuff containers or incompatible materials.

See More Sitagliptin Safety Data Sheet 

Seller Information

Business Type:
Manufactory

Main Products:
Herb Extracts,Cosmetic raw materails,API

Location:
1403,Jinye B Block

Payment Terms:
TT against copy of documents

Average lead Time:
8 days

Total Annual Revenue:
$2.5 million-$5 million

Total Employees:
11-50

Year of Establishment:
2015

Xian ZB Biotech Co.,Ltd is a leading Manufactory supplier of Arbutin, Nicotinamide, Flucytosine based in Xi'an, Shaanxi, China. With a commitment to quality and customer satisfaction, Xian ZB Biotech Co.,Ltd has become a trusted name in the industry. Our product line includes a range of high-quality Arbutin, Nicotinamide, Flucytosine, which are available at competitive prices. Xian ZB Biotech Co.,Ltd has established itself as a reliable supplier of chemical products on the echemi.com.

Inquiry History

2 Inquiries

Country	Product	Purchase Quantity	Date Posted
Oman	Sitagliptin	1 KG	Sep 20, 2026
United States	sitagliptin	1 KG	Sep 14, 2024

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High Purity 99% Sitagliptin Powder CAS 486460-32-6

Product Details

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