Mirogabalin besylate cas 1138245-21-2 in stock
12 Inquiries
1138245-21-2
Analytical Reagent
99%
qingdao
AIRUIKE
1kg
Yes
2024-07-17
api,Intermediates,Organic Chemistry,Inorganic Chemistry,Daily Chemicals,Cosmetic Raw Materals
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Product Description
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Seller Information
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Inquiry History
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DescriptionECHEMI Editorial ReferenceMirogabalin (DS-5565) is a drug developed by Daiichi Sankyo and related to drugs such as gabapentin and pregabalin. Similarly to these drugs, mirogabalin binds to the α2δ calcium channels (1 and 2), but with significantly higher potency than pregabalin. It has shown promising results in Phase II clinical trials for the treatment of diabetic peripheral neuropathic pain, and is currently in Phase III trials.
Mirogabalin besylate (mirogabalin, Tarlige) is a gabapentinoid therapy developed by Daiichi Sankyo, which is approved in Japan for the treatment of postherpetic neuralgia and painful diabetic peripheral neuropathy. Mirogabalin has a potent pain-modulating effect with a unique high affinity and prolonged dissociation rate for the a2delta-1 subunit of voltage-gated calcium (Ca2+) channels (VGCCs) on the dorsal root ganglion resulting in more sustained analgesia compared with traditional gabapentinoids[1].Basic Info-
Product Name:
Mirogabalin besylate
Other Name:Mirogabalin besylate;Mirogabalin besylat;Mirogabalin Besilate;MIROGABALIN BENZENESULFONIC ACID;((1R,5S,6S)-6-(carboxymethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl)methanaminium benzenesulfonate;[(1R,5S,6S)-6-(Aminomethyl)-3-ethylbicyclo[3.2.0] hept-3-en-6-yl]acetic acid benzenesulfonate;2-((1R,5S,6S)-6-(aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl)acetic acid compound with benzenesulfonic acid (1:1);Mirogabalin Besylate 10928
CAS No.:1138245-21-2
Molecular Formula:C18H25NO5S
InChIKeys:OKJXJRVWXYRSAN-QWGAVYBYNA-N
Molecular Weight:367.46
Exact Mass:367.145
Color/Form:White to off-white
Categories:
Characteristics-
PSA:
126.07
XLogP3:4.4968
Critical Temperature & Pressure:Store at -20°C
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Seller Information
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Business Type:
Trader
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Main Products:
api,Intermediates,Organic Chemistry,Inorganic Chemistry,Daily Chemicals,Cosmetic Raw Materals
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Location:
Huangdao District, Qingdao City, Shandong Province (formerly Room 606-2, Building 1, No. 10 Beijing Road, Jiaonan City)
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Payment Terms:
TT against copy of documents,D/P,D/A,TT against B/L draft before shipment,100% TT in advance
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Average lead Time:
15 days
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Total Annual Revenue:
$5 million-$10 million
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Total Employees:
51-100
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Year of Establishment:
2023
Company Certificates-
Credit rating certificate
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Hazardous Chemicals Business License
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Inquiry History12 Inquiries
Country Product Purchase Quantity Date Posted
Pakistan
MIROGABALIN BESYLATE
350 G Feb 10, 2026
Pakistan
Mirogabalin Besilate
1 MT Jul 30, 2025
Pakistan
MIROGABALIN BESYLATE
1 MT Jul 11, 2025
Egypt
Mirogabalin Besylate
250 KG Apr 15, 2026
Pakistan
MIROGABALIN BESYLATE
1 MT Mar 7, 2025
Bangladesh
Mirogabalin Besylate
1 KG Nov 28, 2024
Bangladesh
Mirogabalin Besylate
100 KG Nov 19, 2024
Pakistan
Mirogabalin Besylate
10 KG Sep 4, 2026
Pakistan
Microgabalin Besylate
250 G Aug 19, 2025
Pakistan
MIROGABLIN BESYLATE
350 G Feb 10, 2025
Pakistan
MIROGABALIN BESYLATE
100 KG Oct 31, 2024
Pakistan
Mirogabalin Besylate
1 KG Jul 19, 2024 Post an enquiry for this product