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Home > Encyclopedia > 1,6-Naphthyridin-5(6H)-one,7,8-dihydro-(9CI)

1,6-Naphthyridin-5(6H)-one,7,8-dihydro-(9CI)

1,6-Naphthyridin-5(6H)-one,7,8-dihydro-(9CI) structure

1,6-Naphthyridin-5(6H)-one,7,8-dihydro-(9CI) 

structure
  • CAS No:

    155058-02-9

  • Formula:

    C8H8N2O

  • Chemical Name:

    1,6-Naphthyridin-5(6H)-one,7,8-dihydro-(9CI)

  • Synonyms:

    1,6-Naphthyridin-5(6H)-one,7,8-dihydro-(9CI);7,8-dihydro-1,6-naphthyridin-5(6H)-one;N-methyl-1-(1-methylpiperidin-4-yl)-2-(pyrrolidin-1-yl)ethanamine;1,6-Naphthyridin-5(6H)-one, 7,8-dihydro-;7,8-Dihydro-6H-[1,6]naphthyridin-5-one

  • Categories:

    Pharmaceutical Intermediates  >  Heterocyclic Compound

1,6-Naphthyridin-5(6H)-one,7,8-dihydro-(9CI) Basic Attributes

148.164

148.064

DTXSID50436390

2933990090

Characteristics

42

0.2

1.214±0.06 g/cm3(Predicted)

163-166 °C(Solv: ethyl acetate (141-78-6))

413.9±34.0 °C(Predicted)

1,6-Naphthyridin-5(6H)-one,7,8-dihydro-(9CI) Use and Manufacturing

To a solution of methyl 2-vinylnicotinate (0.40 g, 2.47 mmol, 1 eq) in acetic acid/water 1:1 (4.6 mL), ammonium chloride was added (1.78 g, 33.58 mmol, 14 eq) and the reaction mixture was heated at reflux for 4 h. To a solution of

Computed Properties

Molecular Weight:148.16
XLogP3:0.2
Hydrogen Bond Donor Count:1
Hydrogen Bond Acceptor Count:2
Exact Mass:148.063662883
Monoisotopic Mass:148.063662883
Topological Polar Surface Area:42
Heavy Atom Count:11
Complexity:170
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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