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Flurocitabine

Flurocitabine structure

Flurocitabine 

structure
  • CAS No:

    37717-21-8

  • Formula:

    C9H10FN3O4

  • Chemical Name:

    Flurocitabine

  • Synonyms:

    6H-Furo[2′,3′:4,5]oxazolo[3,2-a]pyrimidine-2-methanol,7-fluoro-2,3,3a,9a-tetrahydro-3-hydroxy-6-imino-,(2R,3R,3aS,9aR)-;6H-Furo[2′,3′:4,5]oxazolo[3,2-a]pyrimidine-2-methanol,7-fluoro-2,3,3a,9a-tetrahydro-3-hydroxy-6-imino-,[2R-(2α,3β,3aβ,9aβ)]-;(2R,3R,3aS,9aR)-7-Fluoro-2,3,3a,9a-tetrahydro-3-hydroxy-6-imino-6H-furo[2′,3′:4,5]oxazolo[3,2-a]pyrimidine-2-methanol;5′-Fluorocyclocytidine;2,2′-Anhydro-1-β-D-arabinofuranosyl-5-fluorocytosine;5-Fluorocyclocytidine;Flurocitabine;Fluorocitabine

  • Categories:

    Biochemical Engineering  >  Saccharides

Description

Flurocitabine is a Cytosine Arabinoside derivative that inhibits pyrimidine synthesis, causing inhibition of DNA synthesis. (NCI)

Flurocitabine Basic Attributes

243.19200

243.19

253-638-9

89TPE33M27

C2343

Characteristics

100.59000

-1.38700

2.11g/cm3

391.7ºC at 760mmHg

190.7ºC

1.813

Drug Information

5-fluoro-2,2'-cyclocytidine

Computed Properties

Molecular Weight:243.19
XLogP3:-2.1
Hydrogen Bond Donor Count:3
Hydrogen Bond Acceptor Count:6
Rotatable Bond Count:1
Exact Mass:243.06553397
Monoisotopic Mass:243.06553397
Topological Polar Surface Area:98.4
Heavy Atom Count:17
Complexity:438
Defined Atom Stereocenter Count:4
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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