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Home > Encyclopedia > 1-(3,4-Diethoxybenzyl)-6,7-diethoxyisoquinoline

1-(3,4-Diethoxybenzyl)-6,7-diethoxyisoquinoline

1-(3,4-Diethoxybenzyl)-6,7-diethoxyisoquinoline structure

1-(3,4-Diethoxybenzyl)-6,7-diethoxyisoquinoline 

structure
  • CAS No:

    486-47-5

  • Formula:

    C24H29NO4

  • Chemical Name:

    1-(3,4-Diethoxybenzyl)-6,7-diethoxyisoquinoline

  • Synonyms:

    Isoquinoline,1-[(3,4-diethoxyphenyl)methyl]-6,7-diethoxy-;Perparine;Isoquinoline,1-(3,4-diethoxybenzyl)-6,7-diethoxy-;1-[(3,4-Diethoxyphenyl)methyl]-6,7-diethoxyisoquinoline;Barbonine;1-(3,4-Diethoxybenzyl)-6,7-diethoxyisoquinoline;6,7-Diethoxy-1-(3,4-diethoxybenzyl)isoquinoline;Ethaverine;Ethylpapaverine;Papaverine,ethyl-;Dyscural;Barbonin;1360-22-1;34487-94-0

Description

Crystals.Insoluble in water; very soluble in hot alcohol; slightly soluble in ether and chloroform.


1-[(3,4-diethoxyphenyl)methyl]-6,7-diethoxyisoquinoline is a member of isoquinolines.

1-(3,4-Diethoxybenzyl)-6,7-diethoxyisoquinoline Basic Attributes

395.496

395.49

207-633-3

2H2HC19DYZ

DTXSID3023009

Characteristics

49.8

5.4

1.1668 (rough estimate)

100 °C

519.44°C (rough estimate)

Drug Information

Agents that inhibit the actions of the parasympathetic nervous system. The major group of drugs used therapeutically for this purpose is the MUSCARINIC ANTAGONISTS. (See all compounds classified as Parasympatholytics.)

Ethaquin

1-(3,4-Diethoxybenzyl)-6,7-diethoxyisoquinoline Use and Manufacturing

Uses

Ethaverine is an analogue of Papaverine (P190500), an antispasmodic. An isoquinoline derivative with the potential for antimicrobial, antimalarial and cytotoxic antiviral agents.

Pharmaceuticals

Computed Properties

Molecular Weight:395.5
XLogP3:5.4
Hydrogen Bond Acceptor Count:5
Rotatable Bond Count:10
Exact Mass:395.20965841
Monoisotopic Mass:395.20965841
Topological Polar Surface Area:49.8
Heavy Atom Count:29
Complexity:462
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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