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14-HYDROXYCODEINE

14-HYDROXYCODEINE structure

14-HYDROXYCODEINE 

structure
  • CAS No:

    4829-46-3

  • Formula:

    C18H21NO4

  • Chemical Name:

    14-HYDROXYCODEINE

  • Synonyms:

    CODEINEIMPF;14-Hydroxycodene;14-HYDROXYCODEINE;3-Methoxy-14-hydroxy-17-methyl-4,5α-epoxymorphinan-7-ene-6α-ol;7,8-Didehydro-4,5α-epoxy-3-methoxy-17-methylmorphinan-6α,14-diol;4,5α-Epoxy-17-methyl-3-methoxy-7,8-didehydromorphinan-6α,14-diol;3-Methoxy-17-methyl-7,8-didehydro-4,5α-epoxymorphinan-6α,14-diol;3-Methoxy-17-methyl-4,5α-epoxy-7,8-didehydromorphinan-6α,14-diol;7,8-DIDEHYDRO-4,5A-EPOXY-3-METHOXY-17-METHYLMORPHINAN-6A,14-DIOL;(5R,6S)-3-Methoxy-17-methyl-7,8-didehydro-4,5-epoxymorphinan-6,14

14-HYDROXYCODEINE Basic Attributes

315.369

315.147064

332OI8E5Z4

DTXSID50197474

Characteristics

62.2

1.03

1.4±0.1 g/cm3

155-157 °C(Solv: benzene (71-43-2); ligroine (8032-32-4))

506.3±50.0 °C at 760 mmHg

260.0±30.1 °C

1.695

Safety Information

P261, P264, P270, P271, P272, P280, P285, P301+P312, P302+P352, P304+P312, P304+P340, P304+P341, P312, P321, P330, P333+P313, P342+P311, P363, P501

H302

|Danger|H302 (100%): Harmful if swallowed [Warning Acute toxicity, oral]|P261, P264, P270, P271, P272, P280, P285, P301+P312, P302+P352, P304+P312, P304+P340, P304+P341, P312, P321, P330, P333+P313, P342+P311, P363, and P501|The GHS information provided by 1 company from 1 notification to the ECHA C&L Inventory.

Drug Information

14-hydroxycodeine

Computed Properties

Molecular Weight:315.4
XLogP3:0.1
Hydrogen Bond Donor Count:2
Hydrogen Bond Acceptor Count:5
Rotatable Bond Count:1
Exact Mass:315.14705815
Monoisotopic Mass:315.14705815
Topological Polar Surface Area:62.2
Heavy Atom Count:23
Complexity:553
Defined Atom Stereocenter Count:5
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

Synthesis Route

1
76-57-3 molecular formula picture

76-57-3

=
+
3
5140-31-8 molecular formula picture

5140-31-8

=

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