Pelitinib(EKB-569)
257933-82-7
99%
2026-10-20
Coenzymes,Inhibito,Enzymes,Zymogens,Substrates,Native Microorganism Creatine Amidinohydrolase
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Product Description
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Seller Information
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DescriptionPelitinib(EKB-569) (CAS No.: 257933-82-7) is supplied by Creative Enzymes, a Manufactory with 6 years on ECHEMI. Key details: content 99%. Contact the supplier on this page to request a quotation or the latest price.ECHEMI Editorial ReferencePelitinib (EKB-569;WAY-EKB 569) is an irreversible inhibitor of EGFR with an IC50 of 38.5 nM; also slightly inhibits Src, MEK/ERK and ErbB2 with IC50s of 282, 800, and 1255 nM, respectively.Basic Info
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Product Name:
Pelitinib
Other Name:2-Butenamide,N-[4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-,(2E)-;(2E)-N-[4-[(3-Chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-2-butenamide;EKB 569;WAY-EKB 569;Pelitinib
CAS No.:257933-82-7
Molecular Formula:C24H23ClFN5O2
InChIKeys:InChIKey=WVUNYSQLFKLYNI-AATRIKPKSA-N
Molecular Weight:467.93
Exact Mass:467.92
EC Number:1312995-182-4
Categories:
Characteristics-
PSA:
90.3
XLogP3:4.5
Appearance:white to beige
Density:1.3±0.1 g/cm3
Melting Point:173-178°C
Boiling Point:655.5°C at 760 mmHg
Flash Point:350.2±31.5 °C
Refractive Index:1.645
Water Solubility:DMSO: soluble5mg/mL, clear (warmed)
Storage Conditions:-20°C Freezer
Vapor Pressure:4.64E-17mmHg at 25°C
Hazard IdentificationClassification of the substance or mixture
Acute toxicity - Category 3, Oral
GHS label elements, including precautionary statements
Pictogram(s) 
Signal word Danger
Hazard statement(s) H301 Toxic if swallowed
Precautionary statement(s) Prevention P264 Wash ... thoroughly after handling.
P270 Do not eat, drink or smoke when using this product.
Response P301+P316 IF SWALLOWED: Get emergency medical help immediately.
P321 Specific treatment (see ... on this label).
P330 Rinse mouth.
Storage P405 Store locked up.
Disposal P501 Dispose of contents/container to an appropriate treatment and disposal facility in accordance with applicable laws and regulations, and product characteristics at time of disposal.
Other hazards which do not result in classification
no data available
Handling and StoragePrecautions for safe handling
Handling in a well ventilated place. Wear suitable protective clothing. Avoid contact with skin and eyes. Avoid formation of dust and aerosols. Use non-sparking tools. Prevent fire caused by electrostatic discharge steam.
Conditions for safe storage, including any incompatibilities
Store the container tightly closed in a dry, cool and well-ventilated place. Store apart from foodstuff containers or incompatible materials.
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Seller Information
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Business Type:
Manufactory
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Main Products:
Coenzymes,Inhibito,Enzymes,Zymogens,Substrates,Native Microorganism Creatine Amidinohydrolase
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Location:
Shirley, New York 11967, USA
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Payment Terms:
TT against copy of documents,D/P
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Average lead Time:
15 days
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Total Annual Revenue:
$1 million-$2.5 million
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Year of Establishment:
2004
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Country Product Purchase Quantity Date Posted Post an enquiry for this product
