Product
Supplier
Encyclopedia
Inquiry
Home > Pharmaceutical Intermediates > Bulk Drug Intermediates > TD-4208 for Sale > Revefenacin CAS 864750-70-9 Long-Acting Muscarinic Antagonist for COPD Maintenance Treatment Research fkhc
Revefenacin CAS 864750-70-9 Long-Acting Muscarinic Antagonist for COPD Maintenance Treatment Research  fkhc buy - large image1
Revefenacin CAS 864750-70-9 Long-Acting Muscarinic Antagonist for COPD Maintenance Treatment Research  fkhc buy - image1
Revefenacin CAS 864750-70-9 Long-Acting Muscarinic Antagonist for COPD Maintenance Treatment Research  fkhc buy - image2
Revefenacin CAS 864750-70-9 Long-Acting Muscarinic Antagonist for COPD Maintenance Treatment Research  fkhc buy - image3
Revefenacin CAS 864750-70-9 Long-Acting Muscarinic Antagonist for COPD Maintenance Treatment Research  fkhc buy - image4
Revefenacin CAS 864750-70-9 Long-Acting Muscarinic Antagonist for COPD Maintenance Treatment Research  fkhc buy - image5
Revefenacin CAS 864750-70-9 Long-Acting Muscarinic Antagonist for COPD Maintenance Treatment Research  fkhc buy - image6

Revefenacin CAS 864750-70-9 Long-Acting Muscarinic Antagonist for COPD Maintenance Treatment Research fkhc

TDS

Unit Price:

$100-130/G FOB

Get Latest Price
CAS No.:

864750-70-9

Grade:

Reagent Grade

Content:

99%

Port:

qingdao

Brand:

//

Packaging:

10mg, 25mg, 50mg, 100mg, 1g

Sample Available:

Yes

Price valid (until):

2026-10-25

Company Type:
Trader
Location:
China
Payment Terms:
TT against copy of documents,TT against B/L draft before shipment,100% TT in advance
Average Lead Time:
7 days
Qualification:
Main Products:

Medetomidine,Medetomidine hydrochloride,D-Lysergic Acid Methyl Ester,SR17018,Fluralaner,GS-441524

  • Product Description

  • Seller Information

  • Description

    —— Product Specification ——

    Parameter Specification Details
    Product Name Revefenacin TD-4208; GSK1160724
    CAS Number 864750-70-9 864750-70-9
    Molecular Formula C₃₅H₄₃N₅O₄ 35 carbons, 43 hydrogens, 5 nitrogens, 4 oxygens
    Molecular Weight 597.75 g/mol —
    Appearance White to off-white solid powder Visual inspection
    Purity ≥98.0% Determined by HPLC
    Ki (M3 receptor) 0.18 nM High affinity at M3 receptor
    Ki (M1/M2/M4/M5) 0.42/0.32/0.56/6.7 nM —
    Solubility DMSO: ≥125 mg/mL (209.12 mM) —
    Storage Powder: -20°C (3 years), 4°C (2 years); In solvent: -80°C (6 months), -20°C (1 month) Protect from light and moisture
    Packaging 5mg, 10mg, 25mg, 50mg, 100mg Amber glass vials
    Application Research use only COPD research, muscarinic receptor studies


    —— Product Detail ——

    Product Overview

    Revefenacin (CAS 864750-70-9), also known as TD-4208 or GSK1160724 and marketed under the brand name Yupelri, is a novel, potent, long-acting, lung-selective inhaled muscarinic antagonist developed by Theravance Biopharma and Mylan . It appears as a white to off-white solid powder with the molecular formula C₃₅H₄₃N₅O₄ and a molecular weight of 597.75 g/mol



    Packaging & Shipping

      • Research quantities: 10mg, 25mg, 50mg amber glass vials

      • Bulk quantities: 100mg, 1g, 5g amber glass bottles

      • Custom packaging available upon request

      • Not classified as hazardous material for transport under normal conditions

      • Product for research and analytical use only; not for human or veterinary use

    Shop CAS 18048-64-1 Eltrombopag Intermediate for Pharmaceutical Research  kr-Detailed Image 1

    — Company profile ——


     Shop CAS 1231930-42-9 Abemaciclib Intermediate for Pharma researech use KR-Detailed Image 1

    Jinan Topfull Chemical Co., Ltd. is an international company rooted in China, specializing in the export of chemical products.

    Our company is committed to making every effort to provide ideal chemical products to potential customers worldwide, including but not limited to: organic/inorganic reagents, biological reagents, plant extracts, pharmaceutical intermediates, active pharmaceutical ingredients (APIs), reference standards, reference substances, peptides, and more. Meanwhile, we have established long-term and stable cooperative relationships with university laboratories and off-campus research institutions, enabling us to offer tailored product services based on customers' actual needs.

    We currently support customized services for most product categories, with supply quantities ranging from milligram (mg), gram (g) to kilogram (kg) levels, as well as wholesale. Product purity covers the full spectrum from 90% to 99.9%, providing customers with one-stop convenient services.

    To date, our products have been exported to developed countries such as the United States, Australia, Canada, Mexico, as well as EU member states including France, Germany, and many other countries and regions such as Nigeria, Ghana, Southeast Asia, and other parts of Asia. Our product quality and services have consistently received high praise.

    Looking ahead, our company will continue to serve as a bridge connecting China and the world, delivering high-quality products and services to global customers.

     

    Shop CAS 1231930-42-9 Abemaciclib Intermediate for Pharma researech use KR-Detailed Image 2

    Shop CAS 1231930-42-9 Abemaciclib Intermediate for Pharma researech use KR-Detailed Image 3

    —— Q&A ——

    Q1: How to confirm the product quality before placing orders?
    A: By sending you available samples. Or if you have special requirements for the goods, we can prepare samples according to your requirements for confirmation.

    Q2: Can you supply free samples?
    A: Yes, we can provide a free sample, but the shipping cost will be paid by the customers. You can either pay the shipping cost or arrange a courier to collect the samples.

    Q3: How do you treat quality complaints?
    A: All our products are strictly tested by our QC and confirmed by QA; unqualified material will not be released to customers. If any quality problem is confirmed to be caused by us, we will replace the goods or refund your payment immediately.

    Q4: What is your MOQ? Is there a discount?
    A: For highvalue products, our MOQ starts from 1g and generally starts from 10g. For other lowprice products, our MOQ starts from 100g and 1kg.
    Q: Is there a discount?
    A: Yes, for larger quantities, we always support with better prices.

    Q5: How to start orders or make payments?
    A: You can send us your Purchase Order (if your company has one), or just send a simple confirmation by email or via Trade Manager. We will then send you a Proforma Invoice with our bank details for your confirmation, and you can make payment accordingly. If you have other preferred payment methods, we are open to discussion and negotiation.



    ECHEMI Editorial Reference
    Revefenacin is a novel biphenyl carbamate tertiary amine agent that belongs to the family of the long-acting muscarinic antagonists (LABA). The labile primary amide in the structure produces a "soft-drug" site that allows rapid systemic clearance and minimizing of the systemically mediated adverse reactions. The LABA group falls into a parent category known as long-acting inhaled bronchodilators and this type of agents are recommended as a maintenance therapy for chronic obstructive pulmonary disease (COPD). From the LABA group, revefenacin is the first once-daily nebulized LAMA treatment. It was developed by Theravance Biopharma and FDA approved on November 9, 2018.|Revefenacin is an Anticholinergic. The mechanism of action of revefenacin is as a Cholinergic Antagonist.|Revefenacin is a synthetic anticholinergic agent that is used as a once daily, nebulized inhalant for maintenance treatment of patients with chronic obstructive pulmonary disease. Revefenacin has not been implicated in causing liver enzyme elevations or clinically apparent acute liver injury.
    Revefenacin is a synthetic anticholinergic that is prescribed for the treatment of chronic obstructive pulmonary disease (COPD).

    Certificates
    • Revefenacin CAS 864750-70-9 Long-Acting Muscarinic Antagonist for COPD Maintenance Treatment Research  fkhc Certificates 1 TDS

    Basic Info
    Product Name:

    TD-4208

    Other Name:

    TD-4208;Revefenacin / TD4208;GSK1160724;CPDD1221;Revefenacin:TD-4208:GSK-1160724;TD 4208;TD4208;1-(2-(4-((4-carbamoylpiperidin-1-yl)methyl)-N-methylbenzamido)ethyl)piperidin-4-yl [1,1'-biphenyl]-2-ylcarbamate;1-[2-[[4-[(4-carbamoylpiperidin-1-yl)methyl]benzoyl]-methylamino]ethyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate

    CAS No.:

    864750-70-9

    Molecular Formula:

    C35H43N5O4

    InChIKeys:

    FYDWDCIFZSGNBU-UHFFFAOYSA-N

    Molecular Weight:

    597.75

    Exact Mass:

    597.75

    UNII:

    G2AE2VE07O

    Color/Form:

    White to off-white

    ATC Code:

    R - Respiratory system

    Characteristics
    PSA:

    108.21

    XLogP3:

    5.4851

    Density:

    1.26±0.1 g/cm3(Predicted)

    Melting Point:

    125 °C

    Boiling Point:

    777.5±60.0 °C(Predicted)

    Water Solubility:

    < 1 mg/ml

    PKA:

    13.34±0.70(Predicted)

    Critical Temperature & Pressure:

    Store at -20°C

  • Seller Information
    Business Type:

    Trader

    Main Products:

    Medetomidine,Medetomidine hydrochloride,D-Lysergic Acid Methyl Ester,SR17018,Fluralaner,GS-441524

    Location:

    RONGSHENG BEIYUANDAJIE 9, LICHENG DISTRICT,JINAN, SHANDONG CHINA

    Payment Terms:

    TT against copy of documents,TT against B/L draft before shipment,100% TT in advance

    Average lead Time:

    7 days

    Total Annual Revenue:

    $1 million-$2.5 million

    Total Employees:

    11-50

    Year of Establishment:

    2022

    Jinan Topfull Chemical Co., Ltd. is a global chemical Industrial and focuses on advanced chemical technology. Specialized in Cosmetic materials, water treatment, fine chemicals and so on. We are looking forward to working together with the people of all circles at home and abroad to seek common development!
  • Country Product Purchase Quantity Date Posted
    Post an enquiry for this product
pic ×

Scan the QR Code to Share

All products displayed on this website are only for non-medical purposes such as industrial applications or scientific research, and cannot be used for clinical diagnosis or treatment of humans or animals. They are not medicinal or edible.

According to relevant laws and regulations and the regulations of this website, units or individuals who purchase hazardous materials should obtain valid qualifications and qualification conditions.

The information shown above is provided by the enterprise itself, and the authenticity, accuracy and legitimacy of the content are the responsibility of the publishing company. ECHEMI does not bear any guarantee responsibility for this. Please be aware that risks in internet transactions objectively exist.

Feedback & Suggestions
Send Message

Thank you for your feedback. If you require further assistance, please contact us by email at info@echemi.com or call us at +86-532-55729510.