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Home > Encyclopedia > 2,6-DIMETHYL-4-(3-NITRO-PHENYL)-PYRIDINE-3,5-DICARBOXYLIC ACID 3-ETHYL ESTER 5-METHYL ESTER

2,6-DIMETHYL-4-(3-NITRO-PHENYL)-PYRIDINE-3,5-DICARBOXYLIC ACID 3-ETHYL ESTER 5-METHYL ESTER

2,6-DIMETHYL-4-(3-NITRO-PHENYL)-PYRIDINE-3,5-DICARBOXYLIC ACID 3-ETHYL ESTER 5-METHYL ESTER structure

2,6-DIMETHYL-4-(3-NITRO-PHENYL)-PYRIDINE-3,5-DICARBOXYLIC ACID 3-ETHYL ESTER 5-METHYL ESTER 

structure
  • CAS No:

    89267-41-4

  • Formula:

    C18H18N2O6

  • Chemical Name:

    2,6-DIMETHYL-4-(3-NITRO-PHENYL)-PYRIDINE-3,5-DICARBOXYLIC ACID 3-ETHYL ESTER 5-METHYL ESTER

  • Synonyms:

    2,6-DIMETHYL-4-(3-NITRO-PHENYL)-PYRIDINE-3,5-DICARBOXYLIC ACID 3-ETHYL ESTER 5-METHYL ESTER;BAY-m 4786;Dehydronitrendipine;Ethyl methyl 2,6-dimethyl-4-(3-nitrophenyl)pyridine-3,5-dicarboxylate;2,6-Dimethyl-4-(3-nitrophenyl)-3,5-pyridinedicarboxylic acid, ethyl methyl ester, hydrochloride

  • Categories:

    Analytical Chemistry  >  Standard

2,6-DIMETHYL-4-(3-NITRO-PHENYL)-PYRIDINE-3,5-DICARBOXYLIC ACID 3-ETHYL ESTER 5-METHYL ESTER Basic Attributes

358.34532

358.116486

DTXSID80237599

Characteristics

111

3.56

1.3±0.1 g/cm3

59-61℃

465.4±45.0 °C at 760 mmHg

235.3±28.7 °C

1.569

Drug Information

Nitrendipine M (dehydro) is a known human metabolite of 3,5-pyridinedicarboxylic acid, 1,4-dihydro-2,6-dimethyl-4-(3-nitrophenyl)-, ethyl methyl ester, (4r)-.

BAY m 4786

2,6-DIMETHYL-4-(3-NITRO-PHENYL)-PYRIDINE-3,5-DICARBOXYLIC ACID 3-ETHYL ESTER 5-METHYL ESTER Use and Manufacturing

Dehydronitrendipine is a derivative of Nitrendipine (N490150), a dihydropyridine calcium channel blocker. Nitrendipine is used in the treatment of primary (essential) hypertension to decrease blood pressure. Antihypertensive.

Computed Properties

Molecular Weight:358.3
XLogP3:3.2
Hydrogen Bond Acceptor Count:7
Rotatable Bond Count:6
Exact Mass:358.11648630
Monoisotopic Mass:358.11648630
Topological Polar Surface Area:111
Heavy Atom Count:26
Complexity:534
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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