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Home > Encyclopedia > 1-(5-Isoquinolinylsulfonyl)piperazine

1-(5-Isoquinolinylsulfonyl)piperazine

1-(5-Isoquinolinylsulfonyl)piperazine structure

1-(5-Isoquinolinylsulfonyl)piperazine 

structure
  • CAS No:

    84468-24-6

  • Formula:

    C13H15N3O2S

  • Chemical Name:

    1-(5-Isoquinolinylsulfonyl)piperazine

  • Synonyms:

    Isoquinoline,5-(1-piperazinylsulfonyl)-;Piperazine,1-(5-isoquinolinylsulfonyl)-;5-(1-Piperazinylsulfonyl)isoquinoline;HA 100 (pharmaceutical);HA 100;1-(5-Isoquinolinylsulfonyl)piperazine

Description

5-(1-piperazinylsulfonyl)isoquinoline is a member of isoquinolines.

1-(5-Isoquinolinylsulfonyl)piperazine Basic Attributes

277.34

277.34

DTXSID60233438

Characteristics

70.7 Ų

162 °C @ Solvent: Ligroine

Safety Information

3

36/37/38

26-36

TM0862600

Xi

|Warning|H315 (100%): Causes skin irritation [Warning Skin corrosion/irritation]|P261, P264, P271, P280, P302+P352, P304+P340, P305+P351+P338, P312, P321, P332+P313, P337+P313, P362, P403+P233, P405, and P501|Aggregated GHS information provided by 38 companies from 1 notifications to the ECHA C&L Inventory. Each notification may be associated with multiple companies.

Drug Information

1-(5-isoquinolinesulfonyl)piperazine

1-(5-Isoquinolinylsulfonyl)piperazine Use and Manufacturing

Exhibited potent inhibition toward protein kinase C and cyclic nucleotide dependent protein kinases

Computed Properties

Molecular Weight:277.34
XLogP3:0.6
Hydrogen Bond Donor Count:1
Hydrogen Bond Acceptor Count:5
Rotatable Bond Count:2
Exact Mass:277.08849790
Monoisotopic Mass:277.08849790
Topological Polar Surface Area:70.7
Heavy Atom Count:19
Complexity:401
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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