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Home > Encyclopedia > (±)-Bunitrolol

(±)-Bunitrolol

(±)-Bunitrolol structure

(±)-Bunitrolol 

structure
  • CAS No:

    34915-68-9

  • Formula:

    C14H20N2O2

  • Chemical Name:

    (±)-Bunitrolol

  • Synonyms:

    Benzonitrile,2-[3-[(1,1-dimethylethyl)amino]-2-hydroxypropoxy]-;2-[3-[(1,1-Dimethylethyl)amino]-2-hydroxypropoxy]benzonitrile;1-tert-Butylamino-3-(2-cyanophenoxy)-2-propanol;1-tert-Butylamino-3-(2-nitrilophenoxy)-2-propanol;Bunitrolol;1-(2-Cyanophenoxy)-2-hydroxy-3-tert-butylaminopropane;dl-Bunitrolol;(±)-Bunitrolol;2-[3-(tert-Butylamino)-2-hydroxypropoxy]benzonitrile;83073-79-4

  • Categories:

    Organic Chemistry  >  Amides

Description

Bunitrolol is an aromatic ether.

(±)-Bunitrolol Basic Attributes

248.326

248.32

DTXSID2022701

2926909090

Characteristics

65.3

2.07698

1.09g/cm3

163-165 °C

414.2ºC at 760mmHg

204.3ºC

Drug Information

bunitrolol

(±)-Bunitrolol Use and Manufacturing

Methods of Manufacturing

It is obtained by the reaction of salicylic nitrile and epoxypropane, and then the ammonolysis of tert-butylamine. Salicylic nitrile is synthesized from salicylaldehyde, first made into oxime, then treated with acetic anhydride and obtained by hydrolysis.

Uses

Beta-blockers. The effect is 4 times stronger than propranolol, and the effect on myocardial inhibition is smaller, about 1/2 of the latter. It is used to treat arrhythmias such as atrial fibrillation, supraventricular tachycardia, angina pectoris and hypertension. Listed in the Federal Republic of Germany in 1985.

Pharmaceuticals

Computed Properties

Molecular Weight:248.32
XLogP3:1.9
Hydrogen Bond Donor Count:2
Hydrogen Bond Acceptor Count:4
Rotatable Bond Count:6
Exact Mass:248.152477885
Monoisotopic Mass:248.152477885
Topological Polar Surface Area:65.3
Heavy Atom Count:18
Complexity:290
Undefined Atom Stereocenter Count:1
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

Material

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