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Home > Encyclopedia > N-(6-(2-(5-bromopyrimidin-2-yloxy)ethoxy)-5-p-tolylpyrimidin-4-yl)-4-(1-hydroxy-2-methylpropan-2-yl)benzenesulfonamide

N-(6-(2-(5-bromopyrimidin-2-yloxy)ethoxy)-5-p-tolylpyrimidin-4-yl)-4-(1-hydroxy-2-methylpropan-2-yl)benzenesulfonamide

N-(6-(2-(5-bromopyrimidin-2-yloxy)ethoxy)-5-p-tolylpyrimidin-4-yl)-4-(1-hydroxy-2-methylpropan-2-yl)benzenesulfonamide structure

N-(6-(2-(5-bromopyrimidin-2-yloxy)ethoxy)-5-p-tolylpyrimidin-4-yl)-4-(1-hydroxy-2-methylpropan-2-yl)benzenesulfonamide 

structure
  • CAS No:

    169679-53-2

  • Formula:

    C27H28BrN5O5S

  • Chemical Name:

    N-(6-(2-(5-bromopyrimidin-2-yloxy)ethoxy)-5-p-tolylpyrimidin-4-yl)-4-(1-hydroxy-2-methylpropan-2-yl)benzenesulfonamide

  • Synonyms:

    N-(6-(2-(5-bromopyrimidin-2-yloxy)ethoxy)-5-p-tolylpyrimidin-4-yl)-4-(1-hydroxy-2-methylpropan-2-yl)benzenesulfonamide;T-0201;Benzenesulfonamide, N-[6-[2-[(5-bromo-2-pyrimidinyl)oxy]ethoxy]-5-(4-methylphenyl)-4-pyrimidinyl]-4-(2-hydroxy-1,1-dimethylethyl)-

N-(6-(2-(5-bromopyrimidin-2-yloxy)ethoxy)-5-p-tolylpyrimidin-4-yl)-4-(1-hydroxy-2-methylpropan-2-yl)benzenesulfonamide Basic Attributes

614.51

613.099

Characteristics

144.8

5.6868

1.455±0.06 g/cm3

179.5-181 °C

753.3±70.0 °C(Predicted)

4.30±0.10

Drug Information

Compounds and drugs that bind to and inhibit or block the activation of ENDOTHELIN RECECPTORS. (See all compounds classified as Endothelin Receptor Antagonists.)

N-(6-2-(5-bromopyrimidin-4-yl)-4-(2-hydroxy-1), 1-dimethylethyl)benzensulfonamide sodium salt sesquihydrate

Computed Properties

Molecular Weight:614.5
XLogP3:4.8
Hydrogen Bond Donor Count:2
Hydrogen Bond Acceptor Count:10
Rotatable Bond Count:11
Exact Mass:613.09945
Monoisotopic Mass:613.09945
Topological Polar Surface Area:145
Heavy Atom Count:39
Complexity:838
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

Synthesis Route

1
245118-89-2 molecular formula picture

245118-89-2

=
2
245118-90-5 molecular formula picture

245118-90-5

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Guide of N-(6-(2-(5-bromopyrimidin-2-yloxy)ethoxy)-5-p-tolylpyrimidin-4-yl)-4-(1-hydroxy-2-methylpropan-2-yl)benzenesulfonamide

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