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Home > Encyclopedia > N-Acetyl-5-aminosalicylic acid

N-Acetyl-5-aminosalicylic acid

N-Acetyl-5-aminosalicylic acid structure

N-Acetyl-5-aminosalicylic acid 

structure
  • CAS No:

    51-59-2

  • Formula:

    C9H9NO4

  • Chemical Name:

    N-Acetyl-5-aminosalicylic acid

  • Synonyms:

    Benzoic acid,5-(acetylamino)-2-hydroxy-;Salicylic acid,5-acetamido-;5-(Acetylamino)-2-hydroxybenzoic acid;5-Acetamidosalicylic acid;5-(Acetylamino)salicylic acid;2-Hydroxy-5-(acetylamino)benzoic acid;N-Acetyl-5-aminosalicylic acid;CJ 46A;2-Hydroxy-5-acetamidobenzoic acid;5-Acetamido-2-hydroxybenzoic acid;3-Carboxyparacetamol;Acetylmesalazine;NSC 54183;858370-63-5

Description

Light-Borwn Cyrstals


N-acetyl-5-aminosalicylic acid is an aminobenzoic acid.

N-Acetyl-5-aminosalicylic acid Basic Attributes

195.17200

195.17

200-107-4

9H126Z3PF5

54183

DTXSID80199002

2924299090

Characteristics

86.63000

1.12180

Light-brown cyrstals

1.462 g/cm3

218 °C

480.2ºC at 760 mmHg

244.2ºC

1.661

Refrigerator

Safety Information

NONH for all modes of transport

26

Hygroscopic

P305 + P351 + P338

H302-H319

|Warning|H302 (100%): Harmful if swallowed [Warning Acute toxicity, oral]|P264, P270, P280, P301+P312, P305+P351+P338, P330, P337+P313, and P501|Aggregated GHS information provided by 39 companies from 2 notifications to the ECHA C&L Inventory. Each notification may be associated with multiple companies.

Drug Information

Mesalazine, N-acetyl is a known human metabolite of mesalazine.

5-acetylaminosalicylate

N-Acetyl-5-aminosalicylic acid Use and Manufacturing

A metabolite of Mesalazine. A Salicylic Acid derivative. Inhibitor of recombinant human thiopurine methyltransferase (hTPMT) A labelled metabolite of Mesalazine. A labelled Salicylic Acid derivative. Inhibitor of recombinant human thiopurine methyltransferase (hTPMT) N-Acetyl Mesalazine is an metabolite of Mesalazine. A Salicylic Acid derivative. Inhibitor of recombinant human thiopurine methyltransferase (hTPMT).

Computed Properties

Molecular Weight:195.17
XLogP3:1.6
Hydrogen Bond Donor Count:3
Hydrogen Bond Acceptor Count:4
Rotatable Bond Count:2
Exact Mass:195.05315777
Monoisotopic Mass:195.05315777
Topological Polar Surface Area:86.6
Heavy Atom Count:14
Complexity:241
Covalently-Bonded Unit Count:1
Compound Is Canonicalized:Yes

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